FUSED POLYCYCLIC COMPOUNDS, COMPOSITIONS, METHODS OF MANUFACTURE AND THEIR USE AS PAF ANTAGONISTS, ANTIHISTAMINES AND/OR ANTIINFLAMMATORY AGENTS - Patent 0412988

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(11)

EP 0 412 988 A1

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(43)	Date of publication:
	20.02.1991 Bulletin 1991/08

(21)	Application number: 89905353.0

(22)	Date of filing: 26.04.1989

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International Patent Classification (IPC):

C07D 209/ 94^{( . )}
A61K 31/ 38^{( . )}
A61K 31/ 40^{( . )}
A61K 31/ 41^{( . )}
A61K 31/ 4184^{( . )}
A61K 31/ 423^{( . )}
A61K 31/ 428^{( . )}
A61K 31/ 44^{( . )}
A61K 31/ 4433^{( . )}
A61K 31/ 454^{( . )}
A61K 31/ 496^{( . )}
A61P 7/ 02^{( . )}
A61P 37/ 08^{( . )}
C07D 209/ 70^{( . )}
C07D 235/ 02^{( . )}
C07D 239/ 70^{( . )}
C07D 249/ 16^{( . )}
C07D 263/ 52^{( . )}
C07D 333/ 80^{( . )}
C07D 401/ 14^{( . )}
C07D 409/ 04^{( . )}
C07D 413/ 04^{( . )}
C07D 417/ 04^{( . )}
C07D 471/ 04^{( . )}
C07D 498/ 04^{( . )}

A61K 31/ 00^{( . )}
A61K 31/ 381^{( . )}
A61K 31/ 403^{( . )}
A61K 31/ 415^{( . )}
A61K 31/ 42^{( . )}
A61K 31/ 425^{( . )}
A61K 31/ 43^{( . )}
A61K 31/ 4427^{( . )}
A61K 31/ 445^{( . )}
A61K 31/ 495^{( . )}
A61K 31/ 53^{( . )}
A61P 29/ 00^{( . )}
A61P 43/ 00^{( . )}
C07D 231/ 54^{( . )}
C07D 237/ 26^{( . )}
C07D 241/ 38^{( . )}
C07D 261/ 20^{( . )}
C07D 277/ 60^{( . )}
C07D 401/ 04^{( . )}
C07D 403/ 04^{( . )}
C07D 409/ 14^{( . )}
C07D 413/ 14^{( . )}
C07D 417/ 14^{( . )}
C07D 495/ 04^{( . )}
C07D 513/ 04^{( . )}

(86)	International application number:
	PCT/US1989/001689

(87)	International publication number:
	WO 1989/010363 (02.11.1989 Gazette 1989/26)

(84)	Designated Contracting States:
	AT BE CH DE FR GB IT LI LU NL SE

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Priority:

28.04.1988 US 19880187105

(71)	Applicant: SCHERING CORPORATION
	Kenilworth, NJ 07030 (US)

(72)	Inventors:
	FRIARY, Richard, J. West Orange, NJ 07052 (US) GREEN, Michael, J. Skillman, NJ 08558 (US) PIWINSKI, John, J. Parsippany, NJ 07054 (US)

(74)	Representative: Ritter, Stephen David, et al
	Mathys & Squire 100 Grays Inn Road London WC1X 8AL London WC1X 8AL (GB)

(54)	FUSED POLYCYCLIC COMPOUNDS, COMPOSITIONS, METHODS OF MANUFACTURE AND THEIR USE AS PAF ANTAGONISTS, ANTIHISTAMINES AND/OR ANTIINFLAMMATORY AGENTS