NOVEL PRODRUG DERIVATIVES OF BIOLOGICALLY ACTIVE AGENTS CONTAINING HYDROXYL GROUPS OR NH-ACIDIC GROUPS - Patent 0454773

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EP 0 454 773 A1

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(43)	Date of publication:
	06.11.1991 Bulletin 1991/45

(21)	Application number: 90902624.0

(22)	Date of filing: 19.01.1990

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International Patent Classification (IPC):

C07D 295/ 08^{( . )}
A61K 31/ 215^{( . )}
A61K 31/ 495^{( . )}
A61K 31/ 535^{( . )}
A61K 47/ 48^{( . )}
C07C 233/ 18^{( . )}
C07C 235/ 06^{( . )}
C07D 233/ 06^{( . )}
C07D 233/ 74^{( . )}
C07D 263/ 58^{( . )}
C07D 295/ 10^{( . )}
C07D 473/ 06^{( . )}
C07D 473/ 18^{( . )}
C07H 17/ 08^{( . )}
C07H 19/ 16^{( . )}
C07J 5/ 00^{( . )}
C07J 43/ 00^{( . )}

A61K 31/ 16^{( . )}
A61K 31/ 24^{( . )}
A61K 31/ 505^{( . )}
A61K 31/ 5375^{( . )}
C07C 229/ 38^{( . )}
C07C 233/ 25^{( . )}
C07C 271/ 22^{( . )}
C07D 233/ 60^{( . )}
C07D 233/ 92^{( . )}
C07D 285/ 135^{( . )}
C07D 295/ 155^{( . )}
C07D 473/ 08^{( . )}
C07D 487/ 04^{( . )}
C07H 19/ 06^{( . )}
C07J 1/ 00^{( . )}
C07J 41/ 00^{( . )}
C07D 285/ 12^{( . )}

(86)	International application number:
	PCT/DK1990/000020

(87)	International publication number:
	WO 1990/008128 (26.07.1990 Gazette 1990/17)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FR GB IT LI LU NL SE

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Priority:

20.01.1989 DK 19890000240

(71)	Applicants:
	Bundgaard, Hans DK-2970 Horsholm (DK) Falch, Erik DK-2950 Vedbaek (DK)

(72)	Inventors:
	Bundgaard, Hans DK-2970 Horsholm (DK) Falch, Erik DK-2950 Vedbaek (DK)

(74)	Representative: Andersen, Henrik Rastrup, et al
	c/o Plougmann & Vingtoft A/S, Sankt Annae Plads 11, P.O. Box 3007 DK-1021 Copenhagen K DK-1021 Copenhagen K (DK)

(54)	NOVEL PRODRUG DERIVATIVES OF BIOLOGICALLY ACTIVE AGENTS CONTAINING HYDROXYL GROUPS OR NH-ACIDIC GROUPS