INHIBITORS OF ASPARTIC PROTEASES - Patent 0538383

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EP 0 538 383 A1

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(43)	Date of publication:
	28.04.1993 Bulletin 1993/17

(21)	Application number: 91913579.0

(22)	Date of filing: 03.07.1991

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International Patent Classification (IPC):

A61K 31/ 16^{( . )}
A61K 31/ 403^{( . )}
A61K 31/ 415^{( . )}
A61K 31/ 66^{( . )}
A61P 31/ 12^{( . )}
C07C 237/ 10^{( . )}
C07C 271/ 22^{( . )}
C07C 317/ 44^{( . )}
C07D 209/ 14^{( . )}
C07D 233/ 61^{( . )}
C07D 295/ 12^{( . )}
C07K 5/ 02^{( . )}
C07K 5/ 065^{( . )}
C07K 14/ 81^{( . )}

A61K 31/ 40^{( . )}
A61K 31/ 404^{( . )}
A61K 31/ 4184^{( . )}
A61K 38/ 55^{( . )}
A61P 43/ 00^{( . )}
C07C 271/ 16^{( . )}
C07C 317/ 28^{( . )}
C07C 323/ 29^{( . )}
C07D 213/ 36^{( . )}
C07D 235/ 08^{( . )}
C07F 9/ 44^{( . )}
C07K 5/ 06^{( . )}
C07K 5/ 072^{( . )}
A61K 38/ 00^{( . )}

(86)	International application number:
	PCT/US1991/004758

(87)	International publication number:
	WO 1992/000956 (23.01.1992 Gazette 1992/03)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FR GB GR IT LI LU NL SE

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Priority:

06.07.1990 US 19900549458

(71)	Applicant: SMITHKLINE BEECHAM CORPORATION
	King of Prussia, PA 19406 (US)

(72)	Inventors:
	DREYER, Geoffrey, Bainbridge Malvern, PA 19355 (US) GLEASON, John, Gerald Downingtown, PA 19335 (US)

(74)	Representative: West, Vivien
	SmithKline Beecham plc Corporate Intellectual Property SB House Great West Road Brentford, Middlesex TW8 9BD Brentford, Middlesex TW8 9BD (GB)

(54)	INHIBITORS OF ASPARTIC PROTEASES