(19)
(11) EP 0 578 745 A1

(12)

(43) Date of publication:
19.01.1994 Bulletin 1994/03

(21) Application number: 92910121.0

(22) Date of filing: 27.03.1992
(51) International Patent Classification (IPC): 
A61K 31/ 415( . )
A61K 31/ 425( . )
A61K 31/ 428( . )
A61K 38/ 00( . )
C07D 213/ 40( . )
C07D 233/ 64( . )
C07D 277/ 22( . )
C07D 409/ 12( . )
C07F 9/ 6574( . )
C07K 14/ 81( . )
A61K 31/ 4184( . )
A61K 31/ 426( . )
A61K 31/ 675( . )
A61P 31/ 12( . )
C07D 213/ 56( . )
C07D 235/ 16( . )
C07D 277/ 62( . )
C07F 9/ 09( . )
C07K 5/ 02( . )
(86) International application number:
PCT/US1992/002238
(87) International publication number:
WO 1992/017490 (15.10.1992 Gazette 1992/26)
(84) Designated Contracting States:
AT BE CH DE DK ES FR GB GR IT LI LU MC NL SE

(30) Priority: 04.04.1991 US 19910679508

(71) Applicant: THE UPJOHN COMPANY
Kalamazoo, Michigan 49001 (US)

(72) Inventors:
  • HESTER, Jackson, B.
    Galesburg, MI 49053 (US)
  • FISHER, Jed, F.
    Three Rivers, MI 49093 (US)
  • THAISRIVONGS, Suvit
    Portage, MI 49002 (US)
  • MAGGIORA, Linda, Louise
    Portage, MI 49002 (US)
  • SAWYER, Tomi, Kim
    Ann Arbor, MI 48108 (US)

(74) Representative: Perry, Robert Edward 
GILL JENNINGS & EVERY Broadgate House 7 Eldon Street
London EC2M 7LH
London EC2M 7LH (GB)

   


(54) PHOSPHORUS CONTAINING COMPOUNDS AS INHIBITORS OF RETROVIRUSES