PEPTIDE ISOTERS CONTAINING A HETEROCYCLE AS H.I.V. INHIBITORS - Patent 0603309

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EP 0 603 309 A1

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(43)	Date of publication:
	29.06.1994 Bulletin 1994/26

(21)	Application number: 92920181.0

(22)	Date of filing: 11.09.1992

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International Patent Classification (IPC):

A61K 31/ 415^{( . )}
A61K 31/ 426^{( . )}
A61P 37/ 04^{( . )}
C07D 233/ 64^{( . )}
C07D 233/ 90^{( . )}
C07D 277/ 20^{( . )}
C07D 277/ 28^{( . )}
C07D 277/ 56^{( . )}
C07D 487/ 04^{( . )}
C07K 14/ 81^{( . )}

A61K 31/ 425^{( . )}
A61P 31/ 12^{( . )}
C07D 233/ 54^{( . )}
C07D 233/ 70^{( . )}
C07D 249/ 08^{( . )}
C07D 277/ 22^{( . )}
C07D 277/ 32^{( . )}
C07D 403/ 06^{( . )}
C07K 5/ 06^{( . )}
C12N 9/ 99^{( . )}

(86)	International application number:
	PCT/US1992/007747

(87)	International publication number:
	WO 1993/005026 (18.03.1993 Gazette 1993/08)

(84)	Designated Contracting States:
	BE CH DE FR GB IT LI NL

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Priority:

11.09.1991 US 19910757751

(71)	Applicant: SMITHKLINE BEECHAM CORPORATION
	Philadelphia Pennsylvania 19101 (US)

(72)	Inventors:
	DREYER, Geoffrey, Bainbridge Malvern, PA 19355 (US) GLEASON, John, Gerald Downingtown, PA 19335 (US) MEEK, Thomas, Downing Saint Davids, PA 19087 (US) THOMPSON, Scott, Kevin Phoenixville, PA 19460 (US)

(74)	Representative: Tocher, Pauline
	SmithKline Beecham plc Corporate Intellectual Property SB House Great West Road Brentford, Middlesex TW8 9BD Brentford, Middlesex TW8 9BD (GB)

(54)	PEPTIDE ISOTERS CONTAINING A HETEROCYCLE AS H.I.V. INHIBITORS