PIPERAZINE AND PIPERIDINE DERIVATIVES, AND THEIR USE AS ANTIPSYCHOTICS - Patent 0625978

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(11)

EP 0 625 978 A1

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(43)	Date of publication:
	30.11.1994 Bulletin 1994/48

(21)	Application number: 93903266.0

(22)	Date of filing: 11.02.1993

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International Patent Classification (IPC):

C07D 333/ 66^{( . )}
A61K 31/ 343^{( . )}
A61K 31/ 403^{( . )}
A61K 31/ 495^{( . )}
A61K 31/ 505^{( . )}
A61P 25/ 00^{( . )}
C07D 261/ 20^{( . )}
C07D 275/ 06^{( . )}
C07D 409/ 12^{( . )}
C07D 413/ 14^{( . )}
C07D 417/ 12^{( . )}
C07D 471/ 04^{( . )}

A61K 31/ 34^{( . )}
A61K 31/ 40^{( . )}
A61K 31/ 404^{( . )}
A61K 31/ 496^{( . )}
A61K 31/ 53^{( . )}
C07D 209/ 40^{( . )}
C07D 275/ 04^{( . )}
C07D 307/ 82^{( . )}
C07D 413/ 12^{( . )}
C07D 417/ 04^{( . )}
C07D 417/ 14^{( . )}
C07D 487/ 04^{( . )}

(86)	International application number:
	PCT/GB1993/000285

(87)	International publication number:
	WO 1993/016073 (19.08.1993 Gazette 1993/20)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

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Priority:

12.02.1992 GB 19920002915

(71)	Applicant: THE WELLCOME FOUNDATION LIMITED
	London NW1 2BP (GB)

(72)	Inventors:
	NORMAN, Mark, Henry Durham, NC 27713 (US) NAVAS, Frank, III Chapel Hill, NC 27516 (US)

(74)	Representative: Stott, Michael John
	The Wellcome Foundation Limited Group Patents & Agreements Langley Court Beckenham Kent BR3 3BS Beckenham Kent BR3 3BS (GB)

(54)	PIPERAZINE AND PIPERIDINE DERIVATIVES, AND THEIR USE AS ANTIPSYCHOTICS