(19)
(11) EP 0 626 847 A1

(12)

(43) Date of publication:
07.12.1994 Bulletin 1994/49

(21) Application number: 93904613.0

(22) Date of filing: 25.01.1993
(51) International Patent Classification (IPC): 
C07D 233/ 64( . )
A61K 38/ 17( . )
A61K 39/ 39( . )
C07D 233/ 00( . )
A61K 31/ 415( . )
A61K 39/ 35( . )
A61P 37/ 00( . )
(86) International application number:
PCT/US1993/000659
(87) International publication number:
WO 1993/014754 (05.08.1993 Gazette 1993/19)
(84) Designated Contracting States:
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 27.01.1992 US 19920826180

(71) Applicants:
  • IMMULOGIC PHARMACEUTICAL CORPORATION
    Waltham, Massachusetts 02154 (US)
  • THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY
    Palo Alto, CA 94304-1850 (US)

(72) Inventors:
  • MELMON, Kenneth L.
    Woodside, CA 94062 (US)
  • GREENSTEIN, Julia L.
    West Newton, MA 02154 (US)
  • KHOSROPOUR, Parisa
    Palo Alto, CA 94303 (US)

(74) Representative: Bizley, Richard Edward, et al 
Hepworth, Lawrence, Bryer & Bizley Merlin House Falconry Court Bakers Lane
Epping Essex CM16 5DQ
Epping Essex CM16 5DQ (GB)

   


(54) HISTAMINE DERIVATIVES AND METHODS FOR THEIR USE AS IMMUNOMODULATORS