<?xml version="1.0" encoding="UTF-8"?><!DOCTYPE ep-patent-document PUBLIC "-//EPO//EP PATENT DOCUMENT 1.4//EN" "ep-patent-document-v1-4.dtd"><ep-patent-document id="EP0636130A1" file="EP93910151NWA1.xml" lang="en" doc-number="0636130" date-publ="19950201" kind="A1" country="EP" status="n" dtd-version="ep-patent-document-v1-4"><SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSE..PTIE..................................................................</B001EP><B003EP>*</B003EP><B007EP>EPregister to ST.36 EBD process v 1.0 kbaumeister@epo.org (15 Jan 2013)</B007EP></eptags></B000><B100><B110>0636130</B110><B130>A1</B130><B140><date>19950201</date></B140><B190>EP</B190></B100><B200><B210>93910151.0</B210><B220><date>19930414</date></B220><B240><B241><date>19941115</date></B241></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>19920008323</B310><B320><date>19920415</date></B320><B330><ctry>GB</ctry></B330><B310>19920016065</B310><B320><date>19920728</date></B320><B330><ctry>GB</ctry></B330><B310>19920019686</B310><B320><date>19920917</date></B320><B330><ctry>GB</ctry></B330><B310>19920026069</B310><B320><date>19921214</date></B320><B330><ctry>GB</ctry></B330></B300><B400><B405><date>19950201</date><bnum>199505</bnum></B405><B430><date>19950201</date><bnum>199505</bnum></B430></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 211/    42            A I                    </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/   415            A I                    </text></classification-ipcr><classification-ipcr sequence="3"><text>A61K  31/  4427            A I                    </text></classification-ipcr><classification-ipcr sequence="4"><text>A61K  31/   443            A I                    </text></classification-ipcr><classification-ipcr sequence="5"><text>A61K  31/  4433            A I                    </text></classification-ipcr><classification-ipcr sequence="6"><text>A61K  31/   445            A I                    </text></classification-ipcr><classification-ipcr sequence="7"><text>A61K  31/   451            A I                    </text></classification-ipcr><classification-ipcr sequence="8"><text>A61P  11/    00            A I                    </text></classification-ipcr><classification-ipcr sequence="9"><text>A61P  11/    08            A I                    </text></classification-ipcr><classification-ipcr sequence="10"><text>C07D 207/    12            A I                    </text></classification-ipcr><classification-ipcr sequence="11"><text>C07D 211/    54            A I                    </text></classification-ipcr><classification-ipcr sequence="12"><text>C07D 401/    06            A I                    </text></classification-ipcr><classification-ipcr sequence="13"><text>C07D 401/    12            A I                    </text></classification-ipcr><classification-ipcr sequence="14"><text>C07D 403/    06            A I                    </text></classification-ipcr><classification-ipcr sequence="15"><text>C07D 405/    06            A I                    </text></classification-ipcr><classification-ipcr sequence="16"><text>C07D 405/    12            A I                    </text></classification-ipcr><classification-ipcr sequence="17"><text>C07D 409/    04            A I                    </text></classification-ipcr><classification-ipcr sequence="18"><text>C07D 409/    06            A I                    </text></classification-ipcr><classification-ipcr sequence="19"><text>C07D 413/    06            A I                    </text></classification-ipcr><classification-ipcr sequence="20"><text>C07D 417/    06            A I                    </text></classification-ipcr></B510EP><B540><B541>en</B541><B542>AZACYCLIC COMPOUNDS</B542><B541>fr</B541><B542>COMPOSES AZACYCLIQUES</B542><B541>de</B541><B542>Azaclyclische Verbindungen</B542></B540></B500><B700><B710><B711><snm>MERCK SHARP &amp; DOHME LTD.</snm><adr><str>Hertford Road</str><city>Hoddesdon Hertfordshire EN11 9NU</city><ctry>GB</ctry></adr></B711></B710><B720><B721><snm>BAKER, Raymond</snm><adr><str>Bulls Cottage, Green Tye</str><city>Much Hadham, Hertfordshire SG10 6JN</city><ctry>GB</ctry></adr></B721><B721><snm>LADDHWAHETTY, Tamara</snm><adr><str>185 Buckhurst Way</str><city>Buckhurst Hill, Essex IG9 6JB</city><ctry>GB</ctry></adr></B721><B721><snm>SEWARD, Eileen Mary</snm><adr><str>15 The Colts, Thorley Park, Bishops Stortford</str><city>Hertfordshire CM23 4DL</city><ctry>GB</ctry></adr></B721><B721><snm>SWAIN, Christopher John</snm><adr><str>8 Mangers Lane</str><city>Duxford, Cambridge CB2 4RN</city><ctry>GB</ctry></adr></B721></B720><B740><B741><snm>Hiscock, Ian James</snm><adr><str>Glaxo Holdings plc, Glaxo House, Berkeley Avenue</str><city>Greenford, Middlesex UB6 0NN</city><ctry>GB</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>CH</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>ES</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>IE</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LU</ctry><ctry>NL</ctry><ctry>PT</ctry><ctry>SE</ctry></B840><B860><B861><dnum><anum>GB1993000788</anum></dnum><date>19930414</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO1993021181</pnum></dnum><date>19931028</date><bnum>199326</bnum></B871></B870></B800></SDOBI></ep-patent-document>