NON-STEROID PROGESTERONE RECEPTOR AGONIST AND ANTAGONIST COMPOUNDS AND METHODS - Patent 0637296

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EP 0 637 296 A1

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(43)	Date of publication:
	08.02.1995 Bulletin 1995/06

(21)	Application number: 93910811.0

(22)	Date of filing: 21.04.1993

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International Patent Classification (IPC):

C07C 25/ 24^{( . )}
C07C 45/ 00^{( . )}
C07C 45/ 68^{( . )}
C07C 47/ 575^{( . )}
C07C 49/ 753^{( . )}
C07C 205/ 06^{( . )}
C07K 14/ 72^{( . )}

C07C 43/ 23^{( . )}
C07C 45/ 67^{( . )}
C07C 45/ 71^{( . )}
C07C 49/ 603^{( . )}
C07C 69/ 017^{( . )}
C07C 205/ 45^{( . )}

(86)	International application number:
	PCT/US1993/003909

(87)	International publication number:
	WO 1993/021145 (28.10.1993 Gazette 1993/26)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

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Priority:

21.04.1992 US 19920872710
16.04.1993 US 19930048646

(71)	Applicants:
	LIGAND PHARMACEUTICALS, INC. San Diego, CA 92121 (US) THE REGENTS OF THE UNIVERSITY OF CALIFORNIA Oakland, California 94612-3550 (US)

(72)	Inventors:
	PATHIRANA, I., Charles San Diego, CA 922128 (US) BERGER, Tina, S. San Diego, CA 91222 (US) STEIN, Robert, S. San Diego, CA 92130 (US) FENICAL, William Del Mar, CA 92130 (US) JONES, Todd, K. Solana Beach, CA 92075 (US) HAMANN, Lawrence, G. San Diego, CA 92122 (US) FARMER, Luc San Diego, CA 92122 (US)

(74)	Representative: Sexton, Jane Helen, et al
	J.A. KEMP & CO. 14 South Square Gray's Inn London WC1R 5LX London WC1R 5LX (GB)

(54)	NON-STEROID PROGESTERONE RECEPTOR AGONIST AND ANTAGONIST COMPOUNDS AND METHODS