(19)
(11) EP 0 639 184 A1

(12)

(43) Date of publication:
22.02.1995 Bulletin 1995/08

(21) Application number: 93910860.0

(22) Date of filing: 28.04.1993
(51) International Patent Classification (IPC): 
C07D 471/ 00( . )
A61K 31/ 517( . )
C07D 239/ 80( . )
C07D 401/ 12( . )
C07D 405/ 12( . )
A61K 31/ 505( . )
A61P 31/ 12( . )
C07D 401/ 06( . )
C07D 403/ 06( . )
(86) International application number:
PCT/US1993/003975
(87) International publication number:
WO 1993/022292 (11.11.1993 Gazette 1993/27)
(84) Designated Contracting States:
AT BE CH DE DK ES FR GB GR IE IT LI LU NL PT SE

(30) Priority: 07.05.1992 US 19920880119
16.12.1992 US 19920991164

(71) Applicant: MERCK & CO. INC.
Rahway New Jersey 07065-0900 (US)

(72) Inventors:
  • LYLE, Terry, A.
    Lederach, PA 19450 (US)
  • TUCKER, Thomas, J.
    North Wales, PA 19454 (US)
  • WISCOUNT, Catherine, M.
    Allentown, PA 18103 (US)

(74) Representative: Thompson, John Dr. 
Merck & Co., Inc. European Patent Department Terlings Park Eastwick Road
Harlow, Essex CM20 2QR
Harlow, Essex CM20 2QR (GB)

   


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