(19)
(11) EP 0 655 066 A1

(12)

(43) Date of publication:
31.05.1995 Bulletin 1995/22

(21) Application number: 93918422.0

(22) Date of filing: 30.07.1993
(51) International Patent Classification (IPC): 
A61K 31/ 40( . )
C07D 498/ 22( . )
C07H 19/ 23( . )
A61P 35/ 00( . )
C07H 9/ 06( . )
(86) International application number:
PCT/US1993/007054
(87) International publication number:
WO 1994/004541 (03.03.1994 Gazette 1994/06)
(84) Designated Contracting States:
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 12.08.1992 US 19920929199

(71) Applicant: THE UPJOHN COMPANY
Kalamazoo, Michigan 49001 (US)

(72) Inventors:
  • ABRAHAM, Irene
    Kalamazoo, MI 49008 (US)
  • ARISTOFF, Paul, A.
    Portage, MI 49002 (US)
  • SKULNICK, Harvey, I.
    Kalamazoo, MI 49009 (US)

(74) Representative: Perry, Robert Edward 
GILL JENNINGS & EVERY Broadgate House 7 Eldon Street
London EC2M 7LH
London EC2M 7LH (GB)

   


(54) PROTEIN KINASE INHIBITORS AND RELATED COMPOUNDS COMBINED WITH TAXOL