(19)
(11)
EP 0 655 066 A1
(12)
(43)
Date of publication:
31.05.1995
Bulletin 1995/22
(21)
Application number:
93918422.0
(22)
Date of filing:
30.07.1993
(51)
International Patent Classification (IPC):
A61K
31/
40
( . )
C07D
498/
22
( . )
C07H
19/
23
( . )
A61P
35/
00
( . )
C07H
9/
06
( . )
(86)
International application number:
PCT/US1993/007054
(87)
International publication number:
WO 1994/004541
(
03.03.1994
Gazette 1994/06)
(84)
Designated Contracting States:
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE
(30)
Priority:
12.08.1992
US 19920929199
(71)
Applicant:
THE UPJOHN COMPANY
Kalamazoo, Michigan 49001 (US)
(72)
Inventors:
ABRAHAM, Irene
Kalamazoo, MI 49008 (US)
ARISTOFF, Paul, A.
Portage, MI 49002 (US)
SKULNICK, Harvey, I.
Kalamazoo, MI 49009 (US)
(74)
Representative:
Perry, Robert Edward
GILL JENNINGS & EVERY Broadgate House 7 Eldon Street
London EC2M 7LH
London EC2M 7LH (GB)
(54)
PROTEIN KINASE INHIBITORS AND RELATED COMPOUNDS COMBINED WITH TAXOL