TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS - Patent 0663827

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EP 0 663 827 A1

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(43)	Date of publication:
	26.07.1995 Bulletin 1995/30

(21)	Application number: 93923134.0

(22)	Date of filing: 27.09.1993

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International Patent Classification (IPC):

A61K 31/ 435^{( . )}
A61K 31/ 443^{( . )}
A61K 31/ 445^{( . )}
A61P 15/ 00^{( . )}
C07D 401/ 12^{( . )}
C07D 409/ 12^{( . )}

A61K 31/ 4427^{( . )}
A61K 31/ 4433^{( . )}
A61P 13/ 02^{( . )}
C07D 221/ 20^{( . )}
C07D 405/ 06^{( . )}
C07D 409/ 14^{( . )}

(86)	International application number:
	PCT/US1993/009152

(87)	International publication number:
	WO 1994/007496 (14.04.1994 Gazette 1994/09)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FR GB GR IE IT LI LU NL PT SE

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Priority:

07.10.1992 US 19920957938

(71)	Applicant: MERCK & CO. INC.
	Rahway New Jersey 07065-0900 (US)

(72)	Inventors:
	EVANS, Ben E. Lansdale, PA 19446 (US) HOBBS, Douglas W. Lansdale, PA 19446 (US) PAWLUCZYK, Joseph M. Warminster, PA 18974 (US) PETTIBONE, Douglas J. Shalfont, PA 18914 (US) RITTLE, Kenneth E. Greenland, PA 18054 (US) RITTLE, Kenneth E. Greenland, PA 18054 (US)

(74)	Representative: Thompson, John Dr., et al
	Merck & Co., Inc. European Patent Department Terlings Park Eastwick Road Harlow, Essex CM20 2QR Harlow, Essex CM20 2QR (GB)

(54)	TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS