<?xml version="1.0" encoding="UTF-8"?><!DOCTYPE ep-patent-document PUBLIC "-//EPO//EP PATENT DOCUMENT 1.4//EN" "ep-patent-document-v1-4.dtd"><ep-patent-document id="EP0663827A1" file="EP93923134NWA1.xml" lang="en" doc-number="0663827" date-publ="19950726" kind="A1" country="EP" status="n" dtd-version="ep-patent-document-v1-4"><SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSE..PTIE..................................................................</B001EP><B003EP>*</B003EP><B007EP>EPregister to ST.36 EBD process v 1.0 kbaumeister@epo.org (15 Jan 2013)</B007EP></eptags></B000><B100><B110>0663827</B110><B130>A1</B130><B140><date>19950726</date></B140><B190>EP</B190></B100><B200><B210>93923134.0</B210><B220><date>19930927</date></B220><B240><B241><date>19950508</date></B241></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>19920957938</B310><B320><date>19921007</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>19950726</date><bnum>199530</bnum></B405><B430><date>19950726</date><bnum>199530</bnum></B430></B400><B500><B510EP><classification-ipcr sequence="1"><text>A61K  31/   435            A I                    </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/  4427            A I                    </text></classification-ipcr><classification-ipcr sequence="3"><text>A61K  31/   443            A I                    </text></classification-ipcr><classification-ipcr sequence="4"><text>A61K  31/  4433            A I                    </text></classification-ipcr><classification-ipcr sequence="5"><text>A61K  31/   445            A I                    </text></classification-ipcr><classification-ipcr sequence="6"><text>A61P  13/    02            A I                    </text></classification-ipcr><classification-ipcr sequence="7"><text>A61P  15/    00            A I                    </text></classification-ipcr><classification-ipcr sequence="8"><text>C07D 221/    20            A I                    </text></classification-ipcr><classification-ipcr sequence="9"><text>C07D 401/    12            A I                    </text></classification-ipcr><classification-ipcr sequence="10"><text>C07D 405/    06            A I                    </text></classification-ipcr><classification-ipcr sequence="11"><text>C07D 409/    12            A I                    </text></classification-ipcr><classification-ipcr sequence="12"><text>C07D 409/    14            A I                    </text></classification-ipcr></B510EP><B540><B541>en</B541><B542>TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS</B542><B541>fr</B541><B542>ANTAGONISTES RECEPTEURS D'OXYTOCINE TOCOLYTIQUE</B542><B541>de</B541><B542>TOKOLYTISCHE OXYTOCINREZEPTORANTAGONISTEN</B542></B540></B500><B700><B710><B711><snm>MERCK &amp; CO. INC.</snm><adr><str>126, East Lincoln Avenue P.O. Box 2000</str><city>Rahway New Jersey 07065-0900</city><ctry>US</ctry></adr></B711></B710><B720><B721><snm>EVANS, Ben E.</snm><adr><str>501 Perkiomen Avenue</str><city>Lansdale, PA 19446</city><ctry>US</ctry></adr></B721><B721><snm>HOBBS, Douglas W.</snm><adr><str>843 Garfield Avenue</str><city>Lansdale, PA 19446</city><ctry>US</ctry></adr></B721><B721><snm>PAWLUCZYK, Joseph M.</snm><adr><str>1264 Emma Lane</str><city>Warminster, PA 18974</city><ctry>US</ctry></adr></B721><B721><snm>PETTIBONE, Douglas J.</snm><adr><str>69 Hickory Lane</str><city>Shalfont, PA 18914</city><ctry>US</ctry></adr></B721><B721><snm>RITTLE, Kenneth E.</snm><adr><str>1955 Old Woods Road</str><city>Greenland, PA 18054</city><ctry>US</ctry></adr></B721><B721><snm>RITTLE, Kenneth E.</snm><adr><str>1955 Old Woods Road</str><city>Greenland, PA 18054</city><ctry>US</ctry></adr></B721></B720><B740><B741><snm>Thompson, John Dr., et al</snm><adr><str>Merck &amp; Co., Inc. European Patent Department Terlings Park Eastwick Road</str><city>Harlow, Essex CM20 2QR</city><ctry>GB</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>CH</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>ES</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>IE</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LU</ctry><ctry>NL</ctry><ctry>PT</ctry><ctry>SE</ctry></B840><B860><B861><dnum><anum>US1993009152</anum></dnum><date>19930927</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO1994007496</pnum></dnum><date>19940414</date><bnum>199409</bnum></B871></B870></B800></SDOBI></ep-patent-document>