(19)
(11) EP 0 665 845 A1

(12)

(43) Date of publication:
09.08.1995 Bulletin 1995/32

(21) Application number: 93923038.0

(22) Date of filing: 21.10.1993
(51) International Patent Classification (IPC): 
C07D 491/ 153( . )
C07D 491/ 22( . )
C07D 491/ 20( . )
C12P 17/ 18( . )
(86) International application number:
PCT/JP1993/001518
(87) International publication number:
WO 1994/009004 (28.04.1994 Gazette 1994/10)
(84) Designated Contracting States:
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 22.10.1992 JP 19920284760

(71) Applicant: THE KITASATO INSTITUTE
Tokyo 108 (JP)

(72) Inventors:
  • OMURA, Satoshi, The Kitasato Institute
    Tokyo 108 (JP)
  • TOMODA, Hiroshi, The Kitasato Institute
    Tokyo 108 (JP)
  • MASUMA, Rokuro, The Kitasato Institute
    Tokyo 108 (JP)

(74) Representative: Woods, Geoffrey Corlett, et al 
J.A. KEMP & CO. 14 South Square Gray's Inn
London WC1R 5LX
London WC1R 5LX (GB)

   


(54) FO-2546 SUBSTANCE, ITS PRODUCTION AND ITS USE AS INHIBITOR OF ACYL-COA CHOLESTEROL ACYLTRANSFERASE