INHIBITORS OF HIV REVERSE TRANSCRIPTASE - Patent 0686148

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EP 0 686 148 A1

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(43)	Date of publication:
	13.12.1995 Bulletin 1995/50

(21)	Application number: 94909663.0

(22)	Date of filing: 15.02.1994

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International Patent Classification (IPC):

A61K 31/ 40^{( . )}
A61K 31/ 403^{( . )}
A61K 31/ 41^{( . )}
A61K 31/ 425^{( . )}
A61K 31/ 4427^{( . )}
A61K 31/ 535^{( . )}
A61P 37/ 04^{( . )}
C07D 209/ 30^{( . )}
C07D 401/ 06^{( . )}
C07D 403/ 12^{( . )}
C07D 405/ 12^{( . )}
C07D 417/ 12^{( . )}

A61K 31/ 4025^{( . )}
A61K 31/ 404^{( . )}
A61K 31/ 42^{( . )}
A61K 31/ 44^{( . )}
A61K 31/ 443^{( . )}
A61P 31/ 12^{( . )}
C07D 209/ 12^{( . )}
C07D 209/ 42^{( . )}
C07D 401/ 12^{( . )}
C07D 405/ 06^{( . )}
C07D 413/ 06^{( . )}
C07D 521/ 00^{( . )}

(86)	International application number:
	PCT/US1994/001694

(87)	International publication number:
	WO 1994/019321 (01.09.1994 Gazette 1994/20)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FR GB GR IE IT LI LU NL PT SE

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Priority:

24.02.1993 US 19930021925

(71)	Applicants:
	MERCK & CO. INC. Rahway New Jersey 07065-0900 (US) Theoharides, Sharon, A. (executrix for the deceased inventor) Landsdale, PA 19446 (US)

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Inventors:

WILLIAMS, Theresa, M.
Harleysville, PA 19438 (US)
CICCARONE, Terrence, M.
East Greenville, PA 18041 (US)
SAARI, Walfred, S.
Lansdale, PA 19446 (US)
WAI, John, S.
Harleysville, PA 19438 (US)
GREENLEE, William, J.
Teaneck, NJ 07666 (US)
BALANI, Suresh, K.
Hatfield, PA 19440 (US)
GOLDMAN, Mark, E.
San Diego, CA 92130 (US)
HOFFMAN, Jacob, M., Jr.
Lansdale, PA 19446 (US)
LUMMA, William, C., Jr.
Pennsburg, PA 18073 (US)
HUFF, Joel, R.
Gwynedd Valley, PA 19437 (US)
ROONEY, Clarence, S.
Worcester, PA 19490 (US)
SANDERSON, Philip, E.
Philadelphia, PA 19118 (US)
THEOHARIDES, Anthony, D. +di
xxx (US)

(74)	Representative: Cole, William Gwyn, et al
	European Patent Department Merck & Co., Inc. Terlings Park Eastwick Road Harlow Essex CM20 2QR Harlow Essex CM20 2QR (GB)

(54)	INHIBITORS OF HIV REVERSE TRANSCRIPTASE