C5a RECEPTOR ANTAGONISTS HAVING SUBSTANTIALLY NO AGONIST ACTIVITY - Patent 0733107

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(11)

EP 0 733 107 A1

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(43)	Date of publication:
	25.09.1996 Bulletin 1996/39

(21)	Application number: 94931155.0

(22)	Date of filing: 16.11.1994

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International Patent Classification (IPC):

G01N 33/ 566^{( . )}
A61K 39/ 395^{( . )}
A61P 1/ 16^{( . )}
A61P 9/ 10^{( . )}
A61P 13/ 02^{( . )}
A61P 17/ 00^{( . )}
A61P 25/ 00^{( . )}
A61P 29/ 00^{( . )}
A61P 37/ 06^{( . )}
C07H 21/ 04^{( . )}
C07K 16/ 18^{( . )}
C12N 1/ 21^{( . )}
C12N 15/ 09^{( . )}
C12P 21/ 02^{( . )}
C12R 1/ 19^{( . )}

A61K 38/ 00^{( . )}
A61P 1/ 00^{( . )}
A61P 9/ 08^{( . )}
A61P 11/ 00^{( . )}
A61P 15/ 00^{( . )}
A61P 19/ 06^{( . )}
A61P 25/ 28^{( . )}
A61P 31/ 04^{( . )}
A61P 43/ 00^{( . )}
C07K 14/ 47^{( . )}
C12N 1/ 19^{( . )}
C12N 5/ 10^{( . )}
C12N 15/ 12^{( . )}
C12P 21/ 08^{( . )}

(86)	International application number:
	PCT/IB1994/000359

(87)	International publication number:
	WO 1995/016033 (15.06.1995 Gazette 1995/25)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

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Priority:

06.12.1993 US 19930162591

(71)	Applicant: CIBA-GEIGY AG
	4002 Basel (CH)

(72)	Inventors:
	VAN OOSTRUM, Jan CH-4112 Flüh (CH) BOYAR, William C. New Providence, NJ 07974 (US) GALAKATOS, Nicholas G. Summit, NJ 07901 (US) PEPPARD, Jane V. Verona, NJ 07044 (US)

(54)	C5a RECEPTOR ANTAGONISTS HAVING SUBSTANTIALLY NO AGONIST ACTIVITY