(19)
(11)
EP 0 737 232 A1
(12)
(43)
Date of publication:
16.10.1996
Bulletin 1996/42
(21)
Application number:
94906465.0
(22)
Date of filing:
28.12.1993
(51)
International Patent Classification (IPC):
G03C
7/
305
( . )
C07C
243/
24
( . )
C07C
245/
00
( . )
C07D
211/
46
( . )
C07D
213/
89
( . )
C07D
239/
54
( . )
C07D
309/
10
( . )
C07D
489/
00
( . )
C07D
491/
08
( . )
C07H
19/
04
( . )
C07K
1/
00
( . )
C07K
5/
00
( . )
C07K
7/
00
( . )
C07K
14/
16
( . )
C08F
20/
52
( . )
C08G
73/
02
( . )
C07B
61/
00
( . )
C07C
243/
40
( . )
C07D
209/
16
( . )
C07D
211/
52
( . )
C07D
239/
46
( . )
C07D
295/
32
( . )
C07D
461/
00
( . )
C07D
489/
02
( . )
C07H
13/
04
( . )
C07H
21/
00
( . )
C07K
1/
04
( . )
C07K
5/
103
( . )
C07K
7/
02
( . )
C08B
37/
00
( . )
C08G
73/
00
( . )
C09D
4/
00
( . )
(86)
International application number:
PCT/US1993/012612
(87)
International publication number:
WO 1995/018186
(
06.07.1995
Gazette 1995/29)
(84)
Designated Contracting States:
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE
(71)
Applicant:
ARQULE, INC.
Medford, MA 02155 (US)
(72)
Inventors:
HOGAN, Joseph, C., Jr.
Belmont, MA 02178 (US)
CASEBIER, David
Hudson, MA 01749 (US)
FURTH, Paul
Waltham, MA 01749 (US)
TU, Cheng
Cambridge, MA 02139 (US)
(74)
Representative:
Lawrence, John
Barker, Brettell & Duncan, 138, Hagley Road, Edgbaston
Birmingham B16 9PW
Birmingham B16 9PW (GB)
(54)
MODULAR DESIGN AND SYNTHESIS OF AMINIMIDE CONTAINING MOLECULES