(19)
(11) EP 0 737 232 A1

(12)

(43) Date of publication:
16.10.1996 Bulletin 1996/42

(21) Application number: 94906465.0

(22) Date of filing: 28.12.1993
(51) International Patent Classification (IPC): 
G03C 7/ 305( . )
C07C 243/ 24( . )
C07C 245/ 00( . )
C07D 211/ 46( . )
C07D 213/ 89( . )
C07D 239/ 54( . )
C07D 309/ 10( . )
C07D 489/ 00( . )
C07D 491/ 08( . )
C07H 19/ 04( . )
C07K 1/ 00( . )
C07K 5/ 00( . )
C07K 7/ 00( . )
C07K 14/ 16( . )
C08F 20/ 52( . )
C08G 73/ 02( . )
C07B 61/ 00( . )
C07C 243/ 40( . )
C07D 209/ 16( . )
C07D 211/ 52( . )
C07D 239/ 46( . )
C07D 295/ 32( . )
C07D 461/ 00( . )
C07D 489/ 02( . )
C07H 13/ 04( . )
C07H 21/ 00( . )
C07K 1/ 04( . )
C07K 5/ 103( . )
C07K 7/ 02( . )
C08B 37/ 00( . )
C08G 73/ 00( . )
C09D 4/ 00( . )
(86) International application number:
PCT/US1993/012612
(87) International publication number:
WO 1995/018186 (06.07.1995 Gazette 1995/29)
(84) Designated Contracting States:
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

(71) Applicant: ARQULE, INC.
Medford, MA 02155 (US)

(72) Inventors:
  • HOGAN, Joseph, C., Jr.
    Belmont, MA 02178 (US)
  • CASEBIER, David
    Hudson, MA 01749 (US)
  • FURTH, Paul
    Waltham, MA 01749 (US)
  • TU, Cheng
    Cambridge, MA 02139 (US)

(74) Representative: Lawrence, John 
Barker, Brettell & Duncan, 138, Hagley Road, Edgbaston
Birmingham B16 9PW
Birmingham B16 9PW (GB)

   


(54) MODULAR DESIGN AND SYNTHESIS OF AMINIMIDE CONTAINING MOLECULES