MODULAR DESIGN AND SYNTHESIS OF OXAZOLONE-DERIVED MOLECULES - Patent 0738155

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(11)

EP 0 738 155 A1

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(43)	Date of publication:
	23.10.1996 Bulletin 1996/43

(21)	Application number: 94907107.0

(22)	Date of filing: 28.12.1993

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International Patent Classification (IPC):

G01N 33/ 545^{( . )}
A61K 31/ 13^{( . )}
A61K 31/ 42^{( . )}
A61K 31/ 695^{( . )}
A61K 38/ 00^{( . )}
A61K 38/ 55^{( . )}
A61K 48/ 00^{( . )}
A61P 25/ 26^{( . )}
A61P 43/ 00^{( . )}
C07C 237/ 22^{( . )}
C07D 211/ 52^{( . )}
C07D 263/ 42^{( . )}
C07D 307/ 54^{( . )}
C07D 333/ 22^{( . )}
C07H 5/ 06^{( . )}
C07H 13/ 04^{( . )}
C07K 1/ 04^{( . )}
C07K 5/ 06^{( . )}
C07K 5/ 103^{( . )}
C08B 37/ 00^{( . )}

A61K 31/ 047^{( . )}
A61K 31/ 165^{( . )}
A61K 31/ 421^{( . )}
A61K 31/ 785^{( . )}
A61K 38/ 46^{( . )}
A61K 47/ 48^{( . )}
A61P 25/ 24^{( . )}
A61P 31/ 04^{( . )}
C07B 61/ 00^{( . )}
C07D 207/ 08^{( . )}
C07D 239/ 47^{( . )}
C07D 265/ 10^{( . )}
C07D 319/ 06^{( . )}
C07D 473/ 34^{( . )}
C07H 7/ 027^{( . )}
C07H 21/ 00^{( . )}
C07K 5/ 02^{( . )}
C07K 5/ 062^{( . )}
C07K 14/ 16^{( . )}
G03C 5/ 30^{( . )}

(86)	International application number:
	PCT/US1993/012591

(87)	International publication number:
	WO 1995/017903 (06.07.1995 Gazette 1995/29)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

(71)	Applicant: ARQULE PARTNERS, L.P.
	Medford, MA 02155 (US)

(72)	Inventors:
	HOGAN, Joseph, C., Jr. Belmont, MA 02178 (US) CASEBIER, David Hudson, MA 01749 (US) FURTH, Paul Waltham, MA 01749 (US) TU, Cheng Cambridge, MA 02139 (US)

(74)	Representative: Lawrence, John, et al
	Barker, Brettell & Duncan, 138, Hagley Road, Edgbaston Birmingham B16 9PW Birmingham B16 9PW (GB)

(54)	MODULAR DESIGN AND SYNTHESIS OF OXAZOLONE-DERIVED MOLECULES