<?xml version="1.0" encoding="UTF-8"?><!DOCTYPE ep-patent-document PUBLIC "-//EPO//EP PATENT DOCUMENT 1.4//EN" "ep-patent-document-v1-4.dtd"><ep-patent-document id="EP0740791A1" file="EP94906537NWA1.xml" lang="en" doc-number="0740791" date-publ="19961106" kind="A1" country="EP" status="n" dtd-version="ep-patent-document-v1-4"><SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIE..................................................................</B001EP><B003EP>*</B003EP><B007EP>EPregister to ST.36 EBD process v 1.0 kbaumeister@epo.org (15 Jan 2013)</B007EP></eptags></B000><B100><B110>0740791</B110><B130>A1</B130><B140><date>19961106</date></B140><B190>EP</B190></B100><B200><B210>94906537.0</B210><B220><date>19940105</date></B220><B240><B241><date>19960726</date></B241></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B400><B405><date>19961106</date><bnum>199645</bnum></B405><B430><date>19961106</date><bnum>199645</bnum></B430></B400><B500><B510EP><classification-ipcr sequence="1"><text>G01N  33/    48            A I                    </text></classification-ipcr><classification-ipcr sequence="2"><text>C07B  61/    00            A I                    </text></classification-ipcr><classification-ipcr sequence="3"><text>C07C 243/    40            A I                    </text></classification-ipcr><classification-ipcr sequence="4"><text>C07D 263/    42            A I                    </text></classification-ipcr><classification-ipcr sequence="5"><text>C07D 265/    10            A I                    </text></classification-ipcr><classification-ipcr sequence="6"><text>C07D 267/    06            A I                    </text></classification-ipcr><classification-ipcr sequence="7"><text>C07D 295/    32            A I                    </text></classification-ipcr><classification-ipcr sequence="8"><text>C07D 307/    54            A I                    </text></classification-ipcr><classification-ipcr sequence="9"><text>C07D 333/    24            A I                    </text></classification-ipcr><classification-ipcr sequence="10"><text>C07D 405/    12            A I                    </text></classification-ipcr><classification-ipcr sequence="11"><text>C07D 409/    12            A I                    </text></classification-ipcr><classification-ipcr sequence="12"><text>C07D 413/    12            A I                    </text></classification-ipcr><classification-ipcr sequence="13"><text>C07K   5/    00            A I                    </text></classification-ipcr><classification-ipcr sequence="14"><text>C07K   7/    00            A I                    </text></classification-ipcr><classification-ipcr sequence="15"><text>C07K  14/    00            A I                    </text></classification-ipcr><classification-ipcr sequence="16"><text>G01N  33/    53            A I                    </text></classification-ipcr><classification-ipcr sequence="17"><text>G01N  33/   566            A I                    </text></classification-ipcr></B510EP><B540><B541>en</B541><B542>SYSTEMATIC MODULAR PRODUCTION OF AMINIMIDE- AND OXAZOLONE-BASED MOLECULES HAVING SELECTED PROPERTIES</B542><B541>fr</B541><B542>PRODUCTION MODULAIRE SYSTEMATIQUE DE MOLECULES A BASE D'AMINIMIDE ET D'OXAZOLONE AYANT DES PROPRIETES CHOISIES</B542><B541>de</B541><B542>SYSTEMATISCHE MODULARE HERSTELLUNG VON AMINIMID- UND OXAZOLONBASIERTEN MOLEKÜLEN MIT AUSGEWÄHLTEN EIGENSCHAFTEN</B542></B540></B500><B700><B710><B711><snm>ARQULE, INC.</snm><adr><str>Suite 3600, 200 Boston Avenue</str><city>Medford, MA 02155</city><ctry>US</ctry></adr></B711></B710><B720><B721><snm>HOGAN, Joseph, C., Jr.</snm><adr><str>50 Oak Avenue</str><city>Belmont, MA 02178</city><ctry>US</ctry></adr></B721></B720><B740><B741><snm>Lawrence, John</snm><adr><str>Barker, Brettell &amp; Duncan, 138, Hagley Road, Edgbaston</str><city>Birmingham B16 9PW</city><ctry>GB</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>CH</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>ES</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>IE</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LU</ctry><ctry>MC</ctry><ctry>NL</ctry><ctry>PT</ctry><ctry>SE</ctry></B840><B860><B861><dnum><anum>US1994000199</anum></dnum><date>19940105</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO1995018972</pnum></dnum><date>19950713</date><bnum>199530</bnum></B871></B870></B800></SDOBI></ep-patent-document>