MALARIAL ASPARTIC PROTEASE INHIBITORS - Patent 0741696

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EP 0 741 696 A1

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(43)	Date of publication:
	13.11.1996 Bulletin 1996/46

(21)	Application number: 95907965.0

(22)	Date of filing: 12.01.1995

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International Patent Classification (IPC):

C07D 295/ 20^{( . )}
A61K 31/ 135^{( . )}
A61K 31/ 415^{( . )}
A61K 31/ 535^{( . )}
A61K 31/ 5375^{( . )}
A61P 33/ 02^{( . )}
C07C 215/ 20^{( . )}
C07C 271/ 16^{( . )}
C07C 271/ 32^{( . )}
C07C 311/ 31^{( . )}
C07C 323/ 58^{( . )}
C07D 233/ 90^{( . )}
C07D 295/ 205^{( . )}
C07D 403/ 12^{( . )}
C07K 5/ 065^{( . )}

A61K 31/ 047^{( . )}
A61K 31/ 165^{( . )}
A61K 31/ 4184^{( . )}
A61K 31/ 5355^{( . )}
A61K 38/ 00^{( . )}
A61P 43/ 00^{( . )}
C07C 233/ 18^{( . )}
C07C 271/ 20^{( . )}
C07C 271/ 40^{( . )}
C07C 317/ 48^{( . )}
C07D 233/ 54^{( . )}
C07D 235/ 24^{( . )}
C07D 307/ 33^{( . )}
C07K 5/ 06^{( . )}
C07K 5/ 078^{( . )}

(86)	International application number:
	PCT/US1995/000017

(87)	International publication number:
	WO 1995/019958 (27.07.1995 Gazette 1995/32)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FR GB GR IE IT LI LU NL PT SE

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Priority:

25.01.1994 US 19940186379

(71)	Applicant: G.D. SEARLE & CO.
	Chicago IL 60680-5110 (US)

(72)	Inventors:
	RUSSELL, Mark, A. Gurnee, IL 60031 (US) MUELLER, Richard, A. Glencoe, IL 60022 (US) BRYANT, Martin, L. Chesterfield, MO 63005 (US) HANSON, Gunnar, H. Skokie, IL 60076 (US)

(74)	Representative: Beil, Hans Christoph, Dr.
	Hansmann & Vogeser, Patent- und Rechtsanwälte, Postfach 80 01 40 65901 Frankfurt 65901 Frankfurt (DE)

(54)	MALARIAL ASPARTIC PROTEASE INHIBITORS