(19)
(11)
EP 0 745 068 A1
(12)
(43)
Date of publication:
04.12.1996
Bulletin 1996/49
(21)
Application number:
95943728.0
(22)
Date of filing:
22.11.1995
(51)
International Patent Classification (IPC):
C07D
249/
02
( . )
A61K
31/
40
( . )
A61K
31/
404
( . )
A61K
31/
415
( . )
A61P
17/
00
( . )
A61P
29/
00
( . )
C07D
207/
32
( . )
C07D
209/
08
( . )
C07D
233/
54
( . )
C07D
233/
58
( . )
C07D
249/
08
( . )
C07F
9/
10
( . )
C07F
9/
6503
( . )
C07F
9/
6515
( . )
A61K
31/
00
( . )
A61K
31/
403
( . )
A61K
31/
41
( . )
A61K
31/
675
( . )
A61P
17/
06
( . )
A61P
35/
00
( . )
C07D
207/
333
( . )
C07D
209/
12
( . )
C07D
233/
56
( . )
C07D
233/
60
( . )
C07D
473/
00
( . )
C07F
9/
572
( . )
C07F
9/
6506
( . )
C07F
9/
6518
( . )
(86)
International application number:
PCT/US1995/016034
(87)
International publication number:
WO 1996/016041
(
30.05.1996
Gazette 1996/25)
(84)
Designated Contracting States:
AT BE CH DE DK ES FR GB GR IE IT LI NL PT SE
(30)
Priority:
22.11.1994
US 19940344282
07.06.1995
US 19950485427
(71)
Applicant:
CLARION PHARMACEUTICALS, INC.
Madison, WI 53711 (US)
(72)
Inventors:
PALTAUF, Friedrich
A-8042 Graz (AT)
HERMETTER, Albin
A-8042 Graz (AT)
FRANZMAIR, Rudolf
A-4040 Linz (AT)
(74)
Representative:
Williams, John Francis
WILLIAMS, POWELL & ASSOCIATES 34 Tavistock Street
London WC2E 7PB
London WC2E 7PB (GB)
(54)
HETEROARYL-SUBSTITUTED DEOXY GLYCERO-PHOSPHOETHANOLAMINES