(19)
(11) EP 0 763 015 A1

(12)

(43) Date of publication:
19.03.1997 Bulletin 1997/12

(21) Application number: 95919869.0

(22) Date of filing: 18.05.1995
(51) International Patent Classification (IPC): 
C07D 295/ 22( . )
C07C 237/ 22( . )
C07C 259/ 00( . )
C07C 275/ 00( . )
C07D 263/ 42( . )
C07D 295/ 32( . )
C07C 233/ 46( . )
C07C 243/ 24( . )
C07C 271/ 00( . )
C07C 327/ 38( . )
C07D 265/ 30( . )
C07D 333/ 24( . )
(86) International application number:
PCT/US1995/006208
(87) International publication number:
WO 1995/032184 (30.11.1995 Gazette 1995/51)
(84) Designated Contracting States:
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 23.05.1994 US 19940248263

(71) Applicant: ARQULE, INC.
Medford, MA 02155 (US)

(72) Inventor:
  • HOGAN, Joseph, C., Jr.
    Belmont, MA 02178 (US)

(74) Representative: Lawrence, John 
Barker, Brettell & Duncan, 138, Hagley Road, Edgbaston
Birmingham B16 9PW
Birmingham B16 9PW (GB)

   


(54) SYSTEMATIC MODULAR PRODUCTION OF AMINIMIDE- AND OXAZOLONE- BASED MOLECULES HAVING AT LEAST TWO STRUCTURAL DIVERSITY ELEMENTS