(19)
(11) EP 0 773 926 A1

(12)

(43) Date of publication:
21.05.1997 Bulletin 1997/21

(21) Application number: 95923745.0

(22) Date of filing: 06.06.1995
(51) International Patent Classification (IPC): 
A61K 31/ 415( . )
A61K 31/ 4402( . )
A61K 31/ 4418( . )
A61K 31/ 47( . )
A61P 31/ 12( . )
C07C 231/ 12( . )
C07C 269/ 06( . )
C07D 213/ 30( . )
C07D 213/ 82( . )
C07D 295/ 185( . )
C07D 295/ 26( . )
C07F 7/ 10( . )
C07K 5/ 062( . )
C07K 5/ 078( . )
A61K 31/ 44( . )
A61K 31/ 4406( . )
A61K 31/ 445( . )
A61K 31/ 535( . )
A61P 43/ 00( . )
C07C 237/ 22( . )
C07C 271/ 22( . )
C07D 213/ 40( . )
C07D 295/ 15( . )
C07D 295/ 192( . )
C07D 521/ 00( . )
C07K 5/ 023( . )
C07K 5/ 065( . )
C07K 5/ 083( . )
(86) International application number:
PCT/US1995/007241
(87) International publication number:
WO 1996/002499 (01.02.1996 Gazette 1996/06)
(84) Designated Contracting States:
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
LT LV SI

(30) Priority: 15.07.1994 US 19940276223

(71) Applicant: MERRELL PHARMACEUTICALS INC.
Cincinnati, Ohio 45215-6300 (US)

(72) Inventors:
  • FARR, Robert, A.
    Loveland, OH 45140 (US)
  • CREGGE, Robert, J.
    Loveland, OH 45140 (US)
  • JANOWICK, David, A.
    Reading, OH 45215 (US)
  • KOHLMAN, Daniel, T.
    Florence, KY 41042 (US)
  • VAN DORSSELAER, Viviane
    F-67100 Strasbourg (FR)
  • SCHIRLIN, Daniel, G.
    F-67450 Lampertheim (FR)
  • TARNUS, Céline
    F-67000 Strasbourg (FR)

(74) Representative: VOSSIUS & PARTNER 
Postfach 86 07 67
81634 München
81634 München (DE)

   


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