| (84) |
Designated Contracting States: |
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AT BE CH DE DK ES FR GB GR IE IT LI LU NL PT SE |
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Designated Extension States: |
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SI |
| (30) |
Priority: |
11.08.1994 US 289474 14.11.1994 US 339369 20.07.1995 US 492461
|
| (43) |
Date of publication of application: |
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28.05.1997 Bulletin 1997/22 |
| (73) |
Proprietor: Merck & Co., Inc. |
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Rahway
New Jersey 07065-0900 (US) |
|
| (72) |
Inventors: |
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- DEUTSCH, Paul, J.
Rahway, NJ 07065 (US)
- EMINI, Emilio, A.
Rahway, NJ 07065 (US)
- VACCA, Joseph, P.
Rahway, NJ 07065 (US)
|
| (74) |
Representative: Cole, William Gwyn et al |
|
European Patent Department,
Merck & Co., Inc.,
Terlings Park,
Eastwick Road Harlow,
Essex CM20 2QR Harlow,
Essex CM20 2QR (GB) |
| (56) |
References cited: :
EP-A- 0 346 847 EP-A- 0 541 168 WO-A-92/08700
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EP-A- 0 486 948 WO-A-92/08698 WO-A-94/14436
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- PROC NATL ACAD SCI, 26 April 1994 USA, pages 4096-4100, VACCA JP; DORSEY BD; SCHLEIF
WA; LEVIN RB; MCDANIEL SL; DARKE PL; ZUGAY J 'L-735,524: an orally bioavailable human
immunodeficiency virus type 1'
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