(19)
(11) EP 0 794 789 A1

(12)

(43) Date of publication:
17.09.1997 Bulletin 1997/38

(21) Application number: 96905380.0

(22) Date of filing: 11.01.1996
(51) International Patent Classification (IPC): 
C07D 277/ 20( . )
A61K 31/ 215( . )
A61K 31/ 421( . )
A61K 31/ 426( . )
A61K 38/ 00( . )
A61P 35/ 00( . )
C07C 323/ 25( . )
C07C 323/ 60( . )
C07D 207/ 34( . )
C07D 215/ 38( . )
C07D 257/ 04( . )
C07D 277/ 38( . )
C07D 307/ 66( . )
C07K 5/ 107( . )
A61K 31/ 195( . )
A61K 31/ 42( . )
A61K 31/ 425( . )
A61K 31/ 44( . )
A61K 38/ 55( . )
A61P 43/ 00( . )
C07C 323/ 59( . )
C07C 329/ 06( . )
C07D 213/ 56( . )
C07D 217/ 22( . )
C07D 263/ 48( . )
C07D 277/ 40( . )
C07K 5/ 103( . )
(86) International application number:
PCT/US1996/001559
(87) International publication number:
WO 1996/021456 (18.07.1996 Gazette 1996/33)
(84) Designated Contracting States:
AT BE CH DE DK ES FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 12.01.1995 US 19950371682
30.05.1995 US 19950451839
03.11.1995 US 19950552554
02.01.1996 US 19960582076

(71) Applicant: UNIVERSITY OF PITTSBURGH
Pittsburgh, Pennsylvania 15260 (US)

(72) Inventors:
  • SEBTI, Said
    Pittsburg, PA 15215 (US)
  • HAMILTON, Andrew
    Pittsburgh, PA 15215 (US)

(74) Representative: Smart, Peter John 
W.H. BECK, GREENER & CO 7 Stone Buildings Lincoln's Inn
London WC2A 3SZ
London WC2A 3SZ (GB)

   


(54) INHIBITORS OF PRENYL TRANSFERASES