(19)
(11) EP 0 807 172 A1

(12)

(43) Date of publication:
19.11.1997 Bulletin 1997/47

(21) Application number: 96903669.0

(22) Date of filing: 24.01.1996
(51) International Patent Classification (IPC): 
C12N 15/ 113( . )
A61K 38/ 00( . )
(86) International application number:
PCT/US1996/001008
(87) International publication number:
WO 1996/023878 (08.08.1996 Gazette 1996/36)
(84) Designated Contracting States:
AT BE CH DE FR GB IE LI LU MC

(30) Priority: 30.01.1995 US 19950380650

(71) Applicants:
  • HYBRIDON, Inc.
    Cambridge, MA 02139 (US)
  • THE WORCESTER FOUNDATION FOR BIOMEDICAL RESEARCH
    Shrewsbury, MA 01545 (US)

(72) Inventors:
  • TEMSAMANI, Jamal
    Worcester, MA 01604 (US)
  • METELEV, Valeri
    Shrewsbury, MA 01545 (US)
  • LEVINA, Asya
    Shrewsbury, MA 01545 (US)
  • AGRAWAL, Sudhir
    Shrewsbury, MA 01545 (US)
  • ZAMECNIK, Paul
    Shrewsbury, MA 01545 (US)

(74) Representative: Vossius, Volker, Dr., et al 
Dr. Volker Vossius, Patentanwaltskanzlei - Rechtsanwaltskanzlei, Holbeinstrasse 5
81679 München
81679 München (DE)

   


(54) HUMAN IMMUNODEFICIENCY VIRUS TRANSCRIPTION INHIBITORS AND METHODS OF THEIR USE