REVERSIBLE PROTEASE INHIBITORS - Patent 0817778

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(11)

EP 0 817 778 A1

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(43)	Date of publication:
	14.01.1998 Bulletin 1998/03

(21)	Application number: 96910499.0

(22)	Date of filing: 21.03.1996

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International Patent Classification (IPC):

C07D 295/ 20^{( . )}
A61K 31/ 535^{( . )}
A61P 43/ 00^{( . )}
C07C 237/ 22^{( . )}
C07D 213/ 72^{( . )}
C07F 7/ 10^{( . )}
C07K 5/ 087^{( . )}
C07K 14/ 81^{( . )}

A61K 31/ 44^{( . )}
A61K 31/ 5375^{( . )}
C07C 231/ 02^{( . )}
C07C 317/ 28^{( . )}
C07D 295/ 215^{( . )}
C07F 9/ 6533^{( . )}
C07K 5/ 107^{( . )}
A61K 38/ 00^{( . )}

(86)	International application number:
	PCT/US1996/003844

(87)	International publication number:
	WO 1996/030353 (03.10.1996 Gazette 1996/44)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

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Priority:

24.03.1995 US 19950409996

(71)	Applicant: ARRIS PHARMACEUTICAL CORPORATION
	South San Francisco, CA 94080 (US)

(72)	Inventors:
	PALMER, James, T. San Ramon, CA 94583 (US) RASNICK, David San Francisco, CA 94110 (US) KLAUS, Jeffrey, L. Burlingame, CA 94010 (US)

(74)	Representative: Baldock, Sharon Claire, et al
	BOULT WADE TENNANT, 27 Furnival Street London EC4A 1PQ London EC4A 1PQ (GB)

(54)	REVERSIBLE PROTEASE INHIBITORS