(19)
(11) EP 0 832 106 A2

(12)

(43) Date of publication:
01.04.1998 Bulletin 1998/14

(21) Application number: 96918098.0

(22) Date of filing: 04.06.1996
(51) International Patent Classification (IPC): 
C07K 7/ 18( . )
A61K 38/ 00( . )
C07K 19/ 00( . )
(86) International application number:
PCT/US1996/008923
(87) International publication number:
WO 1996/039425 (12.12.1996 Gazette 1997/02)
(84) Designated Contracting States:
AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 05.06.1995 US 19950465672
21.05.1996 US 19960647160

(71) Applicants:
  • CORTECH, INC.
    Denver, CO 80221 (US)
  • Cheronis, John C.
    Lakewood, CO 80227 (US)
  • Gyorkos, Albert
    Westminster, CO 80234 (US)
  • Spruce, Lyle W.
    Arvada, CO 8005 (US)
  • Whalley, Eric T.
    Golden, CO 80403 (US)

(72) Inventors:
  • CHERONIS, John, C.
    Lakewood, CO 80227 (US)
  • GYORKOS, Albert
    Westminster, CO 80234 (US)
  • SPRUCE, Lyle, W.
    Arvada, CO 80005 (US)
  • WHALLEY, Eric, T.
    Golden, CO 80403 (US)

(74) Representative: Smart, Peter John 
W.H. BECK, GREENER & CO 7 Stone Buildings Lincoln's Inn
London WC2A 3SZ
London WC2A 3SZ (GB)

   


(54) COMPOUNDS HAVING BRADYKININ ANTAGONISTIC ACTIVITY AND MU-OPIOID AGONISTIC ACTIVITY