(19)
(11) EP 0 833 823 A1

(12)

(43) Date of publication:
08.04.1998 Bulletin 1998/15

(21) Application number: 96913198.0

(22) Date of filing: 26.04.1996
(51) International Patent Classification (IPC): 
C07D( . )
A61K 31/ 38( . )
A61K 31/ 44( . )
A61K 31/ 495( . )
A61K 31/ 55( . )
A61P 3/ 04( . )
C07D 213/ 38( . )
C07D 223/ 08( . )
C07D 239/ 00( . )
C07D 241/ 04( . )
C07D 295/ 096( . )
C07D 309/ 14( . )
C07D 333/ 36( . )
C07D 337/ 04( . )
C07D 401/ 14( . )
C07D 405/ 12( . )
C07D 295/ 02( . )
A61K 31/ 382( . )
A61K 31/ 4402( . )
A61K 31/ 505( . )
A61P 1/ 00( . )
A61P 9/ 12( . )
C07D 213/ 74( . )
C07D 233/ 00( . )
C07D 239/ 42( . )
C07D 295/ 08( . )
C07D 307/ 22( . )
C07D 317/ 58( . )
C07D 335/ 02( . )
C07D 401/ 04( . )
C07D 403/ 04( . )
C07D 409/ 04( . )
(86) International application number:
PCT/US1996/005843
(87) International publication number:
WO 1996/040660 (19.12.1996 Gazette 1997/03)
(84) Designated Contracting States:
AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 07.06.1995 US 19950478383
07.06.1995 US 19950484974
07.11.1995 WO 1995US14472

(71) Applicant: PFIZER INC.
New York, N.Y. 10017 (US)

(72) Inventors:
  • PETERSON, John, M.
    New Haven, CT 06511 (US)
  • BLUM, Charles, A.
    Guilford, CT 06437 (US)
  • CAI, Guolin
    Guilford, CT 06439 (US)
  • HUTCHISON, Alan
    Madison, CT 06443 (US)

(74) Representative: Baillie, Iain Cameron, et al 
c/o Ladas & Parry Altheimer Eck 2
80331 München
80331 München (DE)

   


(54) CERTAIN SUBSTITUTED BENZYLAMINE DERIVATIVES: A NEW CLASS OF NEUROPEPTIDE Y1 SPECIFIC LIGANDS