(19)
(11) EP 0 836 616 A1

(12)

(43) Date of publication:
22.04.1998 Bulletin 1998/17

(21) Application number: 96924886.0

(22) Date of filing: 04.07.1996
(51) International Patent Classification (IPC): 
C12P 21/ 02( . )
A61P 29/ 00( . )
C07D 309/ 10( . )
C07D 491/ 10( . )
C07D 519/ 00( . )
C07K 5/ 062( . )
A61K 38/ 00( . )
C12R 1/ 645( . )
A61K 31/ 495( . )
A61P 37/ 06( . )
C07D 309/ 30( . )
C07D 498/ 08( . )
C07K 5/ 06( . )
C12N 1/ 20( . )
C12R 1/ 465( . )
(86) International application number:
PCT/EP1996/002952
(87) International publication number:
WO 1997/002285 (23.01.1997 Gazette 1997/05)
(84) Designated Contracting States:
AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

(30) Priority: 04.07.1995 GB 19950013596
28.07.1995 GB 19950015495

(71) Applicants:
  • Novartis AG
    4058 Basel (CH)
  • Novartis-Erfindungen Verwaltungsgesellschaft m.b.H.
    1230 Wien (AT)

(72) Inventors:
  • FEHR, Theodor
    CH-4143 Dornach (CH)
  • OBERER, Lukas
    CH-4456 Tenniken (CH)
  • QUESNIAUX RYFFEL, Valerie
    CH-4123 Allschwil (CH)
  • SANGLIER, Jean-Jacques
    CH-4123 Allschwil (CH)
  • SCHULER, Walter
    D-79639 Grenzach-Wyhlen (DE)
  • SEDRANI, Richard
    CH-4054 Basle (CH)

(74) Representative: Roth, Bernhard M., et al 
Novartis AG, Patent- und Markenabteilung, Lichtstrasse 35
4002 Basel
4002 Basel (CH)

   


(54) MACROLIDES