SUBSTITUTED PYRIDYL PYRROLES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE - Patent 0859771

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(11)

EP 0 859 771 A1

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(43)	Date of publication:
	26.08.1998 Bulletin 1998/35

(21)	Application number: 96942022.0

(22)	Date of filing: 30.10.1996

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International Patent Classification (IPC):

A61K 31/ 00^{( . )}
A61K 31/ 4427^{( . )}
A61K 31/ 4433^{( . )}
A61K 31/ 445^{( . )}
A61K 31/ 4523^{( . )}
A61K 31/ 47^{( . )}
A61K 31/ 4725^{( . )}
A61K 31/ 496^{( . )}
A61K 31/ 501^{( . )}
A61K 31/ 506^{( . )}
A61K 31/ 5375^{( . )}
A61P 1/ 00^{( . )}
A61P 3/ 10^{( . )}
A61P 9/ 00^{( . )}
A61P 11/ 00^{( . )}
A61P 29/ 00^{( . )}
A61P 31/ 12^{( . )}
A61P 43/ 00^{( . )}
C07D 401/ 14^{( . )}
C07D 405/ 14^{( . )}
C07D 413/ 14^{( . )}

A61K 31/ 44^{( . )}
A61K 31/ 443^{( . )}
A61K 31/ 4439^{( . )}
A61K 31/ 4465^{( . )}
A61K 31/ 4545^{( . )}
A61K 31/ 472^{( . )}
A61K 31/ 495^{( . )}
A61K 31/ 50^{( . )}
A61K 31/ 505^{( . )}
A61K 31/ 535^{( . )}
A61K 31/ 5377^{( . )}
A61P 3/ 00^{( . )}
A61P 7/ 00^{( . )}
A61P 9/ 10^{( . )}
A61P 19/ 00^{( . )}
A61P 31/ 00^{( . )}
A61P 37/ 00^{( . )}
C07D 401/ 04^{( . )}
C07D 403/ 04^{( . )}
C07D 409/ 14^{( . )}
C07D 417/ 14^{( . )}

(86)	International application number:
	PCT/US1996/018539

(87)	International publication number:
	WO 1997/016442 (09.05.1997 Gazette 1997/20)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

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Priority:

31.10.1995 US 19950007100P
12.03.1996 GB 19960005158
18.04.1996 US 19960015565
10.06.1996 GB 19960012062

(71)	Applicant: MERCK & CO., INC.
	Rahway, New Jersey 07065 (US)

(72)	Inventors:
	de LASZLO, Stephen, E. Rahway, NJ 07065 (US) CHANG, Linda, L. Rahway, NJ 07065 (US) KIM, Dooseop Rahway, NJ 07065 (US) MANTLO, Nathan, B. Rahway, NJ 07065 (US)

(74)	Representative: Thompson, John Dr.
	Merck & Co., Inc. European Patent Department Terlings Park Eastwick Road Harlow, Essex CM20 2QR Harlow, Essex CM20 2QR (GB)

(54)	SUBSTITUTED PYRIDYL PYRROLES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE