(19)
(11) EP 0 861 243 A1

(12)

(43) Date of publication:
02.09.1998 Bulletin 1998/36

(21) Application number: 96931226.0

(22) Date of filing: 18.09.1996
(51) International Patent Classification (IPC): 
A61K 31/ 4025( . )
A61K 31/ 422( . )
A61K 31/ 4439( . )
A61K 31/ 4709( . )
A61K 31/ 498( . )
A61K 31/ 5377( . )
A61P 37/ 08( . )
C07D 215/ 26( . )
C07D 401/ 12( . )
C07D 403/ 12( . )
C07D 409/ 04( . )
C07D 409/ 14( . )
C07D 471/ 04( . )
A61K 31/ 4184( . )
A61K 31/ 437( . )
A61K 31/ 47( . )
A61K 31/ 496( . )
A61K 31/ 517( . )
A61P 29/ 00( . )
A61P 43/ 00( . )
C07D 401/ 04( . )
C07D 401/ 14( . )
C07D 405/ 12( . )
C07D 409/ 12( . )
C07D 413/ 12( . )
C07D 521/ 00( . )
(86) International application number:
PCT/JP1996/002669
(87) International publication number:
WO 1997/011069 (27.03.1997 Gazette 1997/14)
(84) Designated Contracting States:
AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

(30) Priority: 18.09.1995 GB 19950019077

(71) Applicant: FUJISAWA PHARMACEUTICAL CO., LTD.
Osaka-shi Osaka 541 (JP)

(72) Inventors:
  • OKU, Teruo
    Tsukuba-shi, Ibaraki 305 (JP)
  • KAYAKIRI, Hiroshi
    Tsukuba-shi, Ibaraki 305 (JP)
  • ABE, Yoshito
    Inashiki-gun, Ibaraki 300-12 (JP)
  • SAWADA, Yuki
    Tsukuba-shi, Ibaraki 305 (JP)
  • MIZUTANI, Tsuyoshi
    Tsukuba-shi, Ibaraki 305 (JP)

(74) Representative: Türk, Gille, Hrabal, Leifert 
Brucknerstrasse 20
40593 Düsseldorf
40593 Düsseldorf (DE)

   


(54) HETEROCYCLIC COMPOUNDS AS BRADYKININ ANTAGONISTS