(19)
(11)
EP 0 865 427 A1
(12)
(43)
Date of publication:
23.09.1998
Bulletin 1998/39
(21)
Application number:
94922581.0
(22)
Date of filing:
18.07.1994
(51)
International Patent Classification (IPC):
A61K
31/
56
( . )
C07C
401/
00
( . )
A61P
43/
00
( . )
(86)
International application number:
PCT/US1994/008002
(87)
International publication number:
WO 1996/002501
(
01.02.1996
Gazette 1996/06)
(84)
Designated Contracting States:
AT BE CH DE DK ES FR GB GR IE IT LI NL PT SE
(71)
Applicant:
BONE CARE INTERNATIONAL, INC.
Madison, WI 53711 (US)
(72)
Inventors:
MORIARTY, Robert, M.
Oak Park, IL 80302 (US)
GUO, Liang
Bolingbrook, IL 60440 (US)
PENMASTA, Raju, A.
Bolingbrook, IL 60440 (US)
(74)
Representative:
Ford, Michael Frederick, et al
MEWBURN ELLIS York House 23 Kingsway
London WC2B 6HP
London WC2B 6HP (GB)
(54)
SYNTHESIS OF 1ALPHA-HYDROXY VITAMIN D