(19)
(11) EP 0 865 427 A1

(12)

(43) Date of publication:
23.09.1998 Bulletin 1998/39

(21) Application number: 94922581.0

(22) Date of filing: 18.07.1994
(51) International Patent Classification (IPC): 
A61K 31/ 56( . )
C07C 401/ 00( . )
A61P 43/ 00( . )
(86) International application number:
PCT/US1994/008002
(87) International publication number:
WO 1996/002501 (01.02.1996 Gazette 1996/06)
(84) Designated Contracting States:
AT BE CH DE DK ES FR GB GR IE IT LI NL PT SE

(71) Applicant: BONE CARE INTERNATIONAL, INC.
Madison, WI 53711 (US)

(72) Inventors:
  • MORIARTY, Robert, M.
    Oak Park, IL 80302 (US)
  • GUO, Liang
    Bolingbrook, IL 60440 (US)
  • PENMASTA, Raju, A.
    Bolingbrook, IL 60440 (US)

(74) Representative: Ford, Michael Frederick, et al 
MEWBURN ELLIS York House 23 Kingsway
London WC2B 6HP
London WC2B 6HP (GB)

   


(54) SYNTHESIS OF 1ALPHA-HYDROXY VITAMIN D