BENZIMIDZOLYL NEUROPEPTIDE Y RECEPTOR ANTAGONISTS - Patent 0871442

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EP 0 871 442 A1

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(43)	Date of publication:
	21.10.1998 Bulletin 1998/43

(21)	Application number: 97905573.0

(22)	Date of filing: 09.01.1997

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International Patent Classification (IPC):

A61K 31/ 00^{( . )}
A61K 31/ 4184^{( . )}
A61K 31/ 445^{( . )}
A61K 31/ 47^{( . )}
A61K 31/ 4725^{( . )}
A61K 31/ 496^{( . )}
A61K 31/ 506^{( . )}
A61K 31/ 5355^{( . )}
A61K 31/ 5377^{( . )}
C07D 235/ 12^{( . )}
C07D 401/ 12^{( . )}
C07D 403/ 12^{( . )}

A61K 31/ 415^{( . )}
A61K 31/ 4427^{( . )}
A61K 31/ 454^{( . )}
A61K 31/ 472^{( . )}
A61K 31/ 495^{( . )}
A61K 31/ 505^{( . )}
A61K 31/ 535^{( . )}
A61K 31/ 5375^{( . )}
A61P 25/ 04^{( . )}
C07D 401/ 06^{( . )}
C07D 401/ 14^{( . )}
C07D 417/ 14^{( . )}

(86)	International application number:
	PCT/US1997/000511

(87)	International publication number:
	WO 1997/025041 (17.07.1997 Gazette 1997/31)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE
	Designated Extension States:
	RO

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Priority:

09.01.1996 GB 19960000344
12.07.1996 US 19960021636P

(71)	Applicant: ELI LILLY AND COMPANY
	Indianapolis, Indiana 46285 (US)

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Inventors:

ARNOLD, Macklin, B.
Bargersville, IN 46106 (US)
BRITTON, Thomas, C.
Carmel, IN 46033 (US)
BRUNS, Robert, F., Jr.
Carmel, IN 46033 (US)
CANTRELL, Buddy, E.
Fountaintown, IN 46130 (US)
HAPP, Anne, M.
Indianapolis, IN 46220 (US)
HIPSKIND, Philip, A.
New Palestine, IN 46163 (US)
HOWBERT, James, J.
Bellevue, WA 98005 (US)
LOBB, Karen, L.
Indianapolis, IN 46219 (US)
NIXON, James, A.
Indianapolis, IN 46219 (US)
ORNSTEIN, Paul, L.
Carmel, IN 46032 (US)
SMITH, Edward, C.
Indianapolis, IN 46256 (US)
ZARRINMAYEH, Hamideh
Carmel, IN 46032 (US)
ZIMMERMAN, Dennis, M.
Zionsville, IN 46077 (US)

(74)	Representative: Hudson, Christopher Mark
	Lilly Industries Limited European Patent Operations Erl Wood Manor Windlesham Surrey GU20 6PH Windlesham Surrey GU20 6PH (GB)

(54)	BENZIMIDZOLYL NEUROPEPTIDE Y RECEPTOR ANTAGONISTS