ESTERS OF (9-FLUORO-3-METHYL-10-(4-METHYL-1-PIPERAZINYL)-7-OXO-2,3-DIHYDRO-7H-PYRIDO[3,2,1,IJ]-1,3,4-BENZOAXADIAZINE-6-CARBOXYLIC ACID) AND THEIR USE AS ANTIBACTERIAL - Patent 0874633

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EP 0 874 633 A1

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(43)	Date of publication:
	04.11.1998 Bulletin 1998/45

(21)	Application number: 96935143.0

(22)	Date of filing: 31.10.1996

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International Patent Classification (IPC):

A23K 1/ 16^{( . )}
A61K 31/ 535^{( . )}
A61K 31/ 5395^{( . )}
A61P 31/ 04^{( . )}

A61K 31/ 00^{( . )}
A61K 31/ 537^{( . )}
A61P 31/ 00^{( . )}
C07D 498/ 06^{( . )}

(86)	International application number:
	PCT/GB1996/002673

(87)	International publication number:
	WO 1997/025991 (24.07.1997 Gazette 1997/32)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

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Priority:

17.01.1996 GB 19960000888

(71)	Applicant: PFIZER INC.
	New York, N.Y. 10017 (US)

(72)	Inventors:
	DORGAN, Roderick John, Pfizer Limited Sandwich, Kent CT13 9NJ (GB) WEBSTER, Richard Andrew Bentley, Pfizer Limited Sandwich, Kent CT13 9NJ (GB)

(74)	Representative: Stevens, Ian Edward, et al
	Stevens, Hewlett & Perkins, 1 St. Augustine's Place Bristol BS1 4UD Bristol BS1 4UD (GB)

(54)	ESTERS OF (9-FLUORO-3-METHYL-10-(4-METHYL-1-PIPERAZINYL)-7-OXO-2,3-DIHYDRO-7H-PYRIDO[3,2,1,IJ]-1,3,4-BENZOAXADIAZINE-6-CARBOXYLIC ACID) AND THEIR USE AS ANTIBACTERIAL