(19)
(11) EP 0 879 236 A1

(12)

(43) Date of publication:
25.11.1998 Bulletin 1998/48

(21) Application number: 97904193.0

(22) Date of filing: 29.01.1997
(51) International Patent Classification (IPC): 
A01N 43/ 42( . )
A61K 9/ 48( . )
A61K 31/ 44( . )
A61K 47/ 00( . )
C07D 491/ 12( . )
C07D 498/ 14( . )
A61F 13/ 00( . )
A61K 31/ 4375( . )
A61K 31/ 4745( . )
C07D 471/ 14( . )
C07D 491/ 22( . )
(86) International application number:
PCT/US1997/001728
(87) International publication number:
WO 1997/028165 (07.08.1997 Gazette 1997/34)
(84) Designated Contracting States:
AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 30.01.1996 US 19960594235

(60) Divisional application:
07007232.7 / 1829880

(71) Applicant: THE STEHLIN FOUNDATION FOR CANCER RESEARCH
Houston, TX 77002 (US)

(72) Inventors:
  • ZHISONG, Cao
    Friendswood, TX 77546 (US)
  • CIOVANELLA, Beppino, C.
    Houston, TX 77027 (US)

(74) Representative: Kolb, Helga, Dr. Dipl.-Chem., et al 
Hoffmann Eitle, Patent- und Rechtsanwälte, Arabellastrasse 4
81925 München
81925 München (DE)

   


(54) DERIVATIVES OF CAMPTOTHECIN FOR USE IN TREATING CANCER