SYNTHESIS OF CONFORMATIONALLY RESTRICTED AMINO ACIDS, PEPTIDES AND PEPTIDOMIMETICS BY CATALYTIC RING CLOSING METATHESIS - Patent 0880357

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EP 0 880 357 A1

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(43)	Date of publication:
	02.12.1998 Bulletin 1998/49

(21)	Application number: 96919234.0

(22)	Date of filing: 07.06.1996

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International Patent Classification (IPC):

C07K 1/ 04^{( . )}
C07K 7/ 64^{( . )}

C07K 1/ 113^{( . )}

(86)	International application number:
	PCT/US1996/009591

(87)	International publication number:
	WO 1997/026002 (24.07.1997 Gazette 1997/32)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
	Designated Extension States:
	AL LT LV SI

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Priority:

17.01.1996 US 19960010170P

(71)	Applicant: CALIFORNIA INSTITUTE OF TECHNOLOGY
	Pasadena, CA 91125 (US)

(72)	Inventors:
	GRUBBS, Robert, H. South Pasadena, CA 91036 (US) MILLER, J., Scott Wellsley, MA 02181 (US) BLACKWELL, Helen, E. Pasadena, CA 91125 (US)

(74)	Representative: Andrae, Steffen, Dr., et al
	Patentanwälte Andrae Flach Haug Kneissl Bauer Schneider, Balanstrasse 55 81541 München 81541 München (DE)

(54)	SYNTHESIS OF CONFORMATIONALLY RESTRICTED AMINO ACIDS, PEPTIDES AND PEPTIDOMIMETICS BY CATALYTIC RING CLOSING METATHESIS