INTEGRIN RECEPTOR ANTAGONISTS - Patent 0880511

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(11)

EP 0 880 511 A1

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(43)	Date of publication:
	02.12.1998 Bulletin 1998/49

(21)	Application number: 97902931.0

(22)	Date of filing: 13.01.1997

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International Patent Classification (IPC):

C07D 295/ 14^{( . )}
A61K 31/ 4353^{( . )}
A61K 31/ 4375^{( . )}
A61K 31/ 4409^{( . )}
A61K 31/ 4523^{( . )}
A61K 31/ 495^{( . )}
A61P 9/ 10^{( . )}
A61P 43/ 00^{( . )}
C07D 213/ 56^{( . )}
C07D 213/ 73^{( . )}
C07D 213/ 75^{( . )}
C07D 277/ 40^{( . )}
C07D 401/ 12^{( . )}

A61K 31/ 426^{( . )}
A61K 31/ 437^{( . )}
A61K 31/ 44^{( . )}
A61K 31/ 4439^{( . )}
A61K 31/ 4545^{( . )}
A61P 7/ 02^{( . )}
A61P 19/ 08^{( . )}
C07D 213/ 55^{( . )}
C07D 213/ 68^{( . )}
C07D 213/ 74^{( . )}
C07D 277/ 20^{( . )}
C07D 401/ 04^{( . )}
C07D 471/ 04^{( . )}

(86)	International application number:
	PCT/US1997/000572

(87)	International publication number:
	WO 1997/026250 (24.07.1997 Gazette 1997/32)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

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Priority:

16.01.1996 US 19960009965P
16.02.1996 GB 19960003373

(71)	Applicant: MERCK & CO., INC.
	Rahway, New Jersey 07065 (US)

(72)	Inventors:
	HARTMAN, George, D. Rahway, NJ 07065 (US) PERKINS, James, J. Rahway, NJ 07065 (US) DUGGAN, Mark, E. Rahway, NJ 07065 (US) HUNT, Cecilia, A. Rahway, NJ 07065 (US) KRAUSE, Amy, E. Rahway, NJ 07065 (US) IHLE, Nathan, C. Rahway, NJ 07065 (US) ASKEW, Ben Rahway, NJ 07065 (US) HUTCHINSON, John Rahway, NJ 07065 (US) BRASHEAR, Karen Rahway, NJ 07065 (US)

(74)	Representative: Horgan, James Michael Frederic, et al
	Merck & Co., Inc., Terlings Park, Eastwick Road Harlow, Essex CM20 2QR Harlow, Essex CM20 2QR (GB)

(54)	INTEGRIN RECEPTOR ANTAGONISTS