<?xml version="1.0" encoding="UTF-8"?><!DOCTYPE ep-patent-document PUBLIC "-//EPO//EP PATENT DOCUMENT 1.4//EN" "ep-patent-document-v1-4.dtd"><ep-patent-document id="EP0880511A1" file="EP97902931NWA1.xml" lang="en" doc-number="0880511" date-publ="19981202" kind="A1" country="EP" status="n" dtd-version="ep-patent-document-v1-4"><SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSE..PTIE......FI..........................................................</B001EP><B003EP>*</B003EP><B007EP>EPregister to ST.36 EBD process v 1.0 kbaumeister@epo.org (15 Jan 2013)</B007EP></eptags></B000><B100><B110>0880511</B110><B130>A1</B130><B140><date>19981202</date></B140><B190>EP</B190></B100><B200><B210>97902931.0</B210><B220><date>19970113</date></B220><B240><B241><date>19980817</date></B241></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>19960009965P</B310><B320><date>19960116</date></B320><B330><ctry>US</ctry></B330><B310>19960003373</B310><B320><date>19960216</date></B320><B330><ctry>GB</ctry></B330></B300><B400><B405><date>19981202</date><bnum>199849</bnum></B405><B430><date>19981202</date><bnum>199849</bnum></B430></B400><B500><B510EP><classification-ipcr sequence="1"><text>C07D 295/    14            A I                    </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/   426            A I                    </text></classification-ipcr><classification-ipcr sequence="3"><text>A61K  31/  4353            A I                    </text></classification-ipcr><classification-ipcr sequence="4"><text>A61K  31/   437            A I                    </text></classification-ipcr><classification-ipcr sequence="5"><text>A61K  31/  4375            A I                    </text></classification-ipcr><classification-ipcr sequence="6"><text>A61K  31/    44            A I                    </text></classification-ipcr><classification-ipcr sequence="7"><text>A61K  31/  4409            A I                    </text></classification-ipcr><classification-ipcr sequence="8"><text>A61K  31/  4439            A I                    </text></classification-ipcr><classification-ipcr sequence="9"><text>A61K  31/  4523            A I                    </text></classification-ipcr><classification-ipcr sequence="10"><text>A61K  31/  4545            A I                    </text></classification-ipcr><classification-ipcr sequence="11"><text>A61K  31/   495            A I                    </text></classification-ipcr><classification-ipcr sequence="12"><text>A61P   7/    02            A I                    </text></classification-ipcr><classification-ipcr sequence="13"><text>A61P   9/    10            A I                    </text></classification-ipcr><classification-ipcr sequence="14"><text>A61P  19/    08            A I                    </text></classification-ipcr><classification-ipcr sequence="15"><text>A61P  43/    00            A I                    </text></classification-ipcr><classification-ipcr sequence="16"><text>C07D 213/    55            A I                    </text></classification-ipcr><classification-ipcr sequence="17"><text>C07D 213/    56            A I                    </text></classification-ipcr><classification-ipcr sequence="18"><text>C07D 213/    68            A I                    </text></classification-ipcr><classification-ipcr sequence="19"><text>C07D 213/    73            A I                    </text></classification-ipcr><classification-ipcr sequence="20"><text>C07D 213/    74            A I                    </text></classification-ipcr><classification-ipcr sequence="21"><text>C07D 213/    75            A I                    </text></classification-ipcr><classification-ipcr sequence="22"><text>C07D 277/    20            A I                    </text></classification-ipcr><classification-ipcr sequence="23"><text>C07D 277/    40            A I                    </text></classification-ipcr><classification-ipcr sequence="24"><text>C07D 401/    04            A I                    </text></classification-ipcr><classification-ipcr sequence="25"><text>C07D 401/    12            A I                    </text></classification-ipcr><classification-ipcr sequence="26"><text>C07D 471/    04            A I                    </text></classification-ipcr></B510EP><B540><B541>en</B541><B542>INTEGRIN RECEPTOR ANTAGONISTS</B542><B541>fr</B541><B542>ANTAGONISTES DU RECEPTEUR INTEGRINE</B542><B541>de</B541><B542>INTEGRIN-REZEPTOR-ANTAGONISTEN</B542></B540></B500><B700><B710><B711><snm>MERCK &amp; CO., INC.</snm><adr><str>126 East Lincoln Avenue</str><city>Rahway, New Jersey 07065</city><ctry>US</ctry></adr></B711></B710><B720><B721><snm>HARTMAN, George, D.</snm><adr><str>126 East Lincoln Avenue</str><city>Rahway, NJ 07065</city><ctry>US</ctry></adr></B721><B721><snm>PERKINS, James, J.</snm><adr><str>126 East Lincoln Avenue</str><city>Rahway, NJ 07065</city><ctry>US</ctry></adr></B721><B721><snm>DUGGAN, Mark, E.</snm><adr><str>126 East Lincoln Avenue</str><city>Rahway, NJ 07065</city><ctry>US</ctry></adr></B721><B721><snm>HUNT, Cecilia, A.</snm><adr><str>126 East Lincoln Avenue</str><city>Rahway, NJ 07065</city><ctry>US</ctry></adr></B721><B721><snm>KRAUSE, Amy, E.</snm><adr><str>126 East Lincoln Avenue</str><city>Rahway, NJ 07065</city><ctry>US</ctry></adr></B721><B721><snm>IHLE, Nathan, C.</snm><adr><str>126 East Lincoln Avenue</str><city>Rahway, NJ 07065</city><ctry>US</ctry></adr></B721><B721><snm>ASKEW, Ben</snm><adr><str>126 East Lincoln Avenue</str><city>Rahway, NJ 07065</city><ctry>US</ctry></adr></B721><B721><snm>HUTCHINSON, John</snm><adr><str>126 East Lincoln Avenue</str><city>Rahway, NJ 07065</city><ctry>US</ctry></adr></B721><B721><snm>BRASHEAR, Karen</snm><adr><str>126 East Lincoln Avenue</str><city>Rahway, NJ 07065</city><ctry>US</ctry></adr></B721></B720><B740><B741><snm>Horgan, James Michael Frederic, et al</snm><adr><str>Merck &amp; Co., Inc., Terlings Park, Eastwick Road</str><city>Harlow, Essex CM20 2QR</city><ctry>GB</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>CH</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>IE</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LU</ctry><ctry>NL</ctry><ctry>PT</ctry><ctry>SE</ctry></B840><B860><B861><dnum><anum>US1997000572</anum></dnum><date>19970113</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO1997026250</pnum></dnum><date>19970724</date><bnum>199732</bnum></B871></B870></B800></SDOBI></ep-patent-document>