ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE - Patent 0901471

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(11)

EP 0 901 471 A1

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(43)	Date of publication:
	17.03.1999 Bulletin 1999/11

(21)	Application number: 97926600.0

(22)	Date of filing: 16.05.1997

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International Patent Classification (IPC):

A61K 31/ 00^{( . )}
A61K 31/ 4704^{( . )}
A61K 31/ 535^{( . )}
A61K 31/ 5377^{( . )}
A61P 5/ 24^{( . )}
C07D 215/ 22^{( . )}
C07D 215/ 46^{( . )}
C07D 401/ 12^{( . )}
C07D 453/ 02^{( . )}
C07F 7/ 12^{( . )}

A61K 31/ 47^{( . )}
A61K 31/ 4706^{( . )}
A61K 31/ 5375^{( . )}
A61K 31/ 55^{( . )}
A61P 43/ 00^{( . )}
C07D 215/ 36^{( . )}
C07D 401/ 06^{( . )}
C07D 413/ 12^{( . )}
C07D 471/ 08^{( . )}

(86)	International application number:
	PCT/US1997/008479

(87)	International publication number:
	WO 1997/044321 (27.11.1997 Gazette 1997/51)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

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Priority:

20.05.1996 US 19960017150P
10.06.1996 GB 19960012084

(71)	Applicant: MERCK & CO., INC.
	Rahway, New Jersey 07065 (US)

(72)	Inventors:
	GOULET, Mark Rahway, NJ 07065 (US) ALLEN, Eric, E. Rahway, NJ 07065 (US) JIANG, Jinlong Rahway, NJ 07065 (US) SMITH, Roy, G. Rahway, NJ 07065 (US) WALSH, Thomas, F. Rahway, NJ 07065 (US) WYVRATT, Matthew, J., Jr. Rahway, NJ 07065 (US) YANG, Yi, Tien Rahway, NJ 07065 (US) YOUNG, Jonathan, R. Rahway, NJ 07065 (US) DEVITA, Robert, J. Rahway, NJ 07065 (US)

(74)	Representative: Thompson, John Dr., et al
	Merck & Co., Inc. European Patent Department Terlings Park Eastwick Road Harlow, Essex CM20 2QR Harlow, Essex CM20 2QR (GB)

(54)	ANTAGONISTS OF GONADOTROPIN RELEASING HORMONE