<?xml version="1.0" encoding="UTF-8"?><!DOCTYPE ep-patent-document PUBLIC "-//EPO//EP PATENT DOCUMENT 1.4//EN" "ep-patent-document-v1-4.dtd"><ep-patent-document id="EP0904271A1" file="EP96931596NWA1.xml" lang="en" doc-number="0904271" date-publ="19990331" kind="A1" country="EP" status="n" dtd-version="ep-patent-document-v1-4"><SDOBI lang="en"><B000><eptags><B001EP>ATBECHDEDKESFRGBGRITLILUNLSEMCPTIE......FI..........................................................</B001EP><B003EP>*</B003EP><B007EP>EPregister to ST.36 EBD process v 1.0 kbaumeister@epo.org (15 Jan 2013)</B007EP></eptags></B000><B100><B110>0904271</B110><B130>A1</B130><B140><date>19990331</date></B140><B190>EP</B190></B100><B200><B210>96931596.0</B210><B220><date>19960917</date></B220><B240><B241><date>19981026</date></B241></B240><B250>en</B250><B251EP>en</B251EP><B260>en</B260></B200><B300><B310>19960021174P</B310><B320><date>19960501</date></B320><B330><ctry>US</ctry></B330></B300><B400><B405><date>19990331</date><bnum>199913</bnum></B405><B430><date>19990331</date><bnum>199913</bnum></B430></B400><B500><B510EP><classification-ipcr sequence="1"><text>A61K  31/    00            A I                    </text></classification-ipcr><classification-ipcr sequence="2"><text>A61K  31/   505            A I                    </text></classification-ipcr><classification-ipcr sequence="3"><text>A61K  31/   519            A I                    </text></classification-ipcr><classification-ipcr sequence="4"><text>A61K  31/   529            A I                    </text></classification-ipcr><classification-ipcr sequence="5"><text>A61P  35/    00            A I                    </text></classification-ipcr><classification-ipcr sequence="6"><text>C07D 471/    04            A I                    </text></classification-ipcr><classification-ipcr sequence="7"><text>C07K   5/   078            A I                    </text></classification-ipcr><classification-ipcr sequence="8"><text>A61K  38/    00            A N                    </text></classification-ipcr></B510EP><B540><B541>en</B541><B542>5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES</B542><B541>fr</B541><B542>5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES</B542><B541>de</B541><B542>5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINE</B542></B540></B500><B700><B710><B711><snm>THE TRUSTEES OF PRINCETON UNIVERSITY</snm><adr><str>Office of Research &amp; Project Administration, New South Building, 5th Floor, P.O. Box 36</str><city>Princeton, NJ 08544-0036</city><ctry>US</ctry></adr></B711><B711><snm>ELI LILLY AND COMPANY</snm><adr><str>Lilly Corporate Center</str><city>Indianapolis, Indiana 46285</city><ctry>US</ctry></adr></B711></B710><B720><B721><snm>TAYLOR, Edward, C.</snm><adr><str>288 The Western Way</str><city>Princeton, NJ 08540</city><ctry>US</ctry></adr></B721><B721><snm>SHIH, Chuan</snm><adr><str>12532 Pebble Pointe Pass</str><city>Carmel, IN 46033</city><ctry>US</ctry></adr></B721><B721><snm>LEE, Koo</snm><adr><str>9-506 LG Apartment, Doryong-dong, Science Town</str><city>Yusung-gu, Taejon 305-340</city><ctry>KR</ctry></adr></B721><B721><snm>GOSSETT, Lynn, S.</snm><adr><str>5635 North Rural Street</str><city>Indianapolis, IN 46220</city><ctry>US</ctry></adr></B721></B720><B740><B741><snm>Guerre, Dominique, et al</snm><adr><str>Cabinet Germain et Maureau, 12, rue Boileau, BP 6153</str><city>69466 Lyon Cedex 06</city><ctry>FR</ctry></adr></B741></B740></B700><B800><B840><ctry>AT</ctry><ctry>BE</ctry><ctry>CH</ctry><ctry>DE</ctry><ctry>DK</ctry><ctry>ES</ctry><ctry>FI</ctry><ctry>FR</ctry><ctry>GB</ctry><ctry>GR</ctry><ctry>IE</ctry><ctry>IT</ctry><ctry>LI</ctry><ctry>LU</ctry><ctry>MC</ctry><ctry>NL</ctry><ctry>PT</ctry><ctry>SE</ctry></B840><B860><B861><dnum><anum>US1996014822</anum></dnum><date>19960917</date></B861><B862>en</B862></B860><B870><B871><dnum><pnum>WO1997041115</pnum></dnum><date>19971106</date><bnum>199747</bnum></B871></B870></B800></SDOBI></ep-patent-document>