HIV PROTEASE INHIBITORS USEFUL FOR THE TREATMENT OF AIDS - Patent 0912170

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EP 0 912 170 A1

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(43)	Date of publication:
	06.05.1999 Bulletin 1999/18

(21)	Application number: 97923431.0

(22)	Date of filing: 29.04.1997

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International Patent Classification (IPC):

A61K 31/ 00^{( . )}
A61K 31/ 365^{( . )}
A61K 31/ 496^{( . )}
A61K 31/ 5375^{( . )}
A61P 31/ 18^{( . )}
C07C 237/ 22^{( . )}
C07D 207/ 26^{( . )}
C07D 295/ 185^{( . )}
C07D 307/ 93^{( . )}
C07D 405/ 06^{( . )}

A61K 31/ 165^{( . )}
A61K 31/ 495^{( . )}
A61K 31/ 535^{( . )}
A61P 31/ 00^{( . )}
C07C 233/ 66^{( . )}
C07C 311/ 18^{( . )}
C07D 241/ 04^{( . )}
C07D 303/ 36^{( . )}
C07D 401/ 06^{( . )}

(86)	International application number:
	PCT/US1997/006595

(87)	International publication number:
	WO 1997/040825 (06.11.1997 Gazette 1997/47)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

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Priority:

02.05.1996 US 19960016685P
27.06.1996 GB 19960013488

(71)	Applicant: MERCK & CO., INC.
	Rahway, New Jersey 07065 (US)

(72)	Inventors:
	HUNGATE, Randall, W. Rahway, NJ 07065 (US) KIM, Byeong, Moon Rahway, NJ 07065 (US) VACCA, Joseph, P. Rahway, NJ 07065 (US)

(74)	Representative: Horgan, James Michael Frederic, et al
	Merck & Co., Inc., Terlings Park, Eastwick Road Harlow, Essex CM20 2QR Harlow, Essex CM20 2QR (GB)

(54)	HIV PROTEASE INHIBITORS USEFUL FOR THE TREATMENT OF AIDS