(19)
(11) EP 0 934 293 A1

(12)

(43) Date of publication:
11.08.1999 Bulletin 1999/32

(21) Application number: 97937066.0

(22) Date of filing: 30.07.1997
(51) International Patent Classification (IPC): 
C07D 295/ 20( . )
A61K 31/ 496( . )
A61P 11/ 06( . )
A61P 43/ 00( . )
C07D 213/ 56( . )
C07D 233/ 14( . )
C07D 233/ 64( . )
C07D 239/ 42( . )
C07D 401/ 12( . )
A61K 31/ 495( . )
A61K 31/ 506( . )
A61P 29/ 00( . )
C07D 211/ 26( . )
C07D 213/ 70( . )
C07D 233/ 26( . )
C07D 239/ 22( . )
C07D 295/ 215( . )
(86) International application number:
PCT/US1997/013422
(87) International publication number:
WO 1998/004537 (05.02.1998 Gazette 1998/05)
(84) Designated Contracting States:
AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 30.07.1996 US 19960023139P
17.07.1997 US 19970895772

(71) Applicant: ARRIS PHARMACEUTICAL CORPORATION
South San Francisco, CA 94080 (US)

(72) Inventors:
  • DENER, Jeffrey, Mark
    Daly City, CA 94015 (US)
  • KUO, Elaine, Yee-Lin
    Berkeley, CA 94709 (US)
  • RICE, Ken, Duane
    Sausalito, CA 94965 (US)
  • WANG, Vivian, Rueywen
    Redwood City, CA 94065 (US)
  • YOUNG, Wendy, Beth
    San Mateo, CA 94403 (US)

(74) Representative: Thomson, Paul Anthony, et al 
Potts, Kerr & Co. 15, Hamilton Square
Birkenhead Merseyside L41 6BR
Birkenhead Merseyside L41 6BR (GB)

   


(54) NOVEL COMPOUNDS AND COMPOSITIONS FOR TREATING DISEASES ASSOCIATED WITH TRYPTASE ACTIVITY