INTEGRIN ANTAGONISTS - Patent 0934305

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(11)

EP 0 934 305 A1

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(43)	Date of publication:
	11.08.1999 Bulletin 1999/32

(21)	Application number: 97938568.0

(22)	Date of filing: 25.08.1997

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International Patent Classification (IPC):

A61K 31/ 4375^{( . )}
A61K 31/ 454^{( . )}
A61K 31/ 4709^{( . )}
A61K 31/ 506^{( . )}
A61P 3/ 14^{( . )}
A61P 9/ 10^{( . )}
A61P 27/ 02^{( . )}
A61P 35/ 00^{( . )}
C07D 471/ 04^{( . )}
C07K 5/ 02^{( . )}

A61K 31/ 444^{( . )}
A61K 31/ 4545^{( . )}
A61K 31/ 497^{( . )}
A61P 3/ 10^{( . )}
A61P 9/ 08^{( . )}
A61P 19/ 10^{( . )}
A61P 29/ 02^{( . )}
A61P 43/ 00^{( . )}
C07D 519/ 00^{( . )}
A61K 38/ 00^{( . )}

(86)	International application number:
	PCT/US1997/014912

(87)	International publication number:
	WO 1998/008840 (05.03.1998 Gazette 1998/09)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

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Priority:

29.08.1996 US 19960025123P
19.12.1996 US 19960033579P
13.02.1997 GB 19970003015
20.05.1997 US 19970047177P

(71)	Applicant: MERCK & CO., INC.
	Rahway, New Jersey 07065 (US)

(72)	Inventors:
	DUGGAN, Mark, E. Rahway, NJ 07065 (US) HARTMAN, George, D. Rahway, NJ 07065 (US) HOFFMAN, William, F. Rahway, NJ 07065 (US) MEISSNER, Robert, S. Rahway, NJ 07065 (US) PERKINS, James, J. Rahway, NJ 07065 (US) ASKEW, Ben, C. Rahway, NJ 07065 (US) COLEMAN, Paul, J. Rahway, NJ 07065 (US) HUTCHINSON, John, H. Rahway, NJ 07065 (US) NAYLOR-OLSEN, Adel, M. Rahway, NJ 07065 (US)

(74)	Representative: Horgan, James Michael Frederic, et al
	Merck & Co., Inc., Terlings Park, Eastwick Road Harlow, Essex CM20 2QR Harlow, Essex CM20 2QR (GB)

(54)	INTEGRIN ANTAGONISTS