(19)
(11)
EP 0 939 758 A1
(12)
(43)
Date of publication:
08.09.1999
Bulletin 1999/36
(21)
Application number:
97911690.0
(22)
Date of filing:
10.10.1997
(51)
International Patent Classification (IPC):
C07D
413/
14
( . )
C07D
417/
14
( . )
C07K
5/
06
( . )
A61K
38/
00
( . )
C07D
417/
12
( . )
C07F
5/
02
( . )
C07K
5/
097
( . )
(86)
International application number:
PCT/US1997/018410
(87)
International publication number:
WO 1998/016524
(
23.04.1998
Gazette 1998/16)
(84)
Designated Contracting States:
AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
(30)
Priority:
11.10.1996
US 19960731384
11.10.1996
US 19960036257P
(71)
Applicant:
COR THERAPEUTICS, INC.
South San Francisco, CA 94080 (US)
(72)
Inventors:
ZHU, Bing-Yan
Foster City, CA 94404 (US)
SCARBOROUGH, Robert, M.
Belmont, CA 94002 (US)
(74)
Representative:
Mouget-Goniot, Claire, et al
Cabinet Orès, 6, Avenue de Messine
75008 Paris
75008 Paris (FR)
(54)
HETEROCYCLIC DERIVATIVES AS FACTOR Xa INHIBITORS