BENZODIAZEPINE HYDRAZIDE DERIVATIVES AS INHIBITORS OF HIV INTEGRASE - Patent 0949926

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EP 0 949 926 A1

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(43)	Date of publication:
	20.10.1999 Bulletin 1999/42

(21)	Application number: 97911906.0

(22)	Date of filing: 27.10.1997

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International Patent Classification (IPC):

A61K 31/ 5513^{( . )}
C07D 403/ 12^{( . )}

C07D 243/ 20^{( . )}

(86)	International application number:
	PCT/US1997/019230

(87)	International publication number:
	WO 1998/018473 (07.05.1998 Gazette 1998/18)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FI FR GB GR IE IT LI LU NL PT SE

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Priority:

31.10.1996 US 19960029348P
22.11.1996 GB 19960024375

(71)	Applicant: MERCK & CO., INC.
	Rahway, New Jersey 07065 (US)

(72)	Inventors:
	BELL, Ian, M. Rahway, NJ 07065 (US) GUARE, James, P., Jr. Rahway, NJ 07065 (US) HAZUDA, Daria, Jean Rahway, NJ 07065 (US) MUNSON, Peter, M. Rahway, NJ 07065 (US) THOMPSON, Wayne, J. Rahway, NJ 07065 (US) VACCA, Joseph, P. Rahway, NJ 07065 (US)

(74)	Representative: Thompson, John Dr., et al
	Merck & Co., Inc. European Patent Department Terlings Park Eastwick Road Harlow, Essex CM20 2QR Harlow, Essex CM20 2QR (GB)

(54)	BENZODIAZEPINE HYDRAZIDE DERIVATIVES AS INHIBITORS OF HIV INTEGRASE