(19)
(11) EP 0 954 315 A2

(12)

(43) Date of publication:
10.11.1999 Bulletin 1999/45

(21) Application number: 97941542.0

(22) Date of filing: 11.09.1997
(51) International Patent Classification (IPC): 
A61K 9/ 00( . )
A61K 47/ 00( . )
A61K 47/ 06( . )
A61K 47/ 12( . )
A61K 31/ 517( . )
C07D 239/ 94( . )
A61K 47/ 10( . )
A61K 47/ 14( . )
(86) International application number:
PCT/US1997/016145
(87) International publication number:
WO 1998/010767 (19.03.1998 Gazette 1998/11)
(84) Designated Contracting States:
AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 13.09.1996 US 19960026067P
20.11.1996 US 19960031436P
08.01.1997 US 19970034981P
03.06.1997 US 19970048372P

(71) Applicant: Sugen, Inc.
South San Francisco, CA 94080 (US)

(72) Inventors:
  • McMAHON, Gerald
    Kenwood, CA 95452 (US)
  • SHAWVER, Laura, Kay
    San Francisco, CA 94112 (US)
  • NAROG, Blair
    Sunnydale, CA 94086 (US)
  • TANG, Peng, Cho
    Moraga, CA 94556 (US)
  • HIRTH, Klaus, Peter
    San Francisco, CA 94114 (US)

(74) Representative: Moon, Donald Keith, et al 
BREWER & SON Quality House Quality Court Chancery Lane
London WC2A 1HT
London WC2A 1HT (GB)

   


(54) USE OF QUINAZOLINE DERIVATIVES FOR THE MANUFACTURE OF A MEDICAMENT IN THE TREATMENT OF HYPERPROLIFERATIVE SKIN DISORDERS