POLYPROLYL INHIBITORS OF CYCLOPHILIN

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EP 0 966 479 A1

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(43)	Date of publication:
	29.12.1999 Bulletin 1999/52

(21)	Application number: 97953231.0

(22)	Date of filing: 08.12.1997

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International Patent Classification (IPC):

A61K 45/ 00^{( . )}
A61K 38/ 08^{( . )}
A61P 25/ 00^{( . )}
A61P 25/ 28^{( . )}
C07K 7/ 06^{( . )}

A61K 38/ 07^{( . )}
A61K 38/ 55^{( . )}
A61P 25/ 16^{( . )}
C07K 5/ 10^{( . )}

(86)	International application number:
	PCT/US1997/023102

(87)	International publication number:
	WO 1998/025950 (18.06.1998 Gazette 1998/24)

(84)	Designated Contracting States:
	AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

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Priority:

09.12.1996 US 19960761902

(71)	Applicant: GUILFORD PHARMACEUTICALS INC.
	Baltimore, Maryland 21224 (US)

(72)	Inventors:
	HAMILTON, Gregory, S. Catonsville, MD 21228 (US) WEI, Ling Lutherville, MD 21093 (US) STEINER, Joseph, P. Hampstead, MD 21074 (US)

(74)	Representative: Kihn, Pierre Emile Joseph, et al
	Office de Brevets Ernest T. Freylinger 234, route d'Arlon B.P. 48 8001 Strassen 8001 Strassen (LU)

(54)	POLYPROLYL INHIBITORS OF CYCLOPHILIN