(19)
(11) EP 0 971 896 A1

(12)

(43) Date of publication:
19.01.2000 Bulletin 2000/03

(21) Application number: 98919133.3

(22) Date of filing: 24.03.1998
(51) International Patent Classification (IPC)7C07D 215/48, A61K 31/47, C07B 57/00
(86) International application number:
PCT/EP9801/700
(87) International publication number:
WO 9842/673 (01.10.1998 Gazette 1998/39)
(84) Designated Contracting States:
AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE
Designated Extension States:
AL LT LV MK RO SI

(30) Priority: 26.03.1997 GB 9706294

(71) Applicant: GLAXO WELLCOME S.p.A.
37100 Verona (IT)

(72) Inventors:
  • DI FABIO, Romano,Glaxo Wellcome S.p.A.
    I-37100 Verona (IT)
  • BERTANI, Barbara,Glaxo Wellcome S.p.A.
    I-37100 Verona (IT)
  • ALVARO, Giuseppe,Glaxo Wellcome S.p.A.
    I-37100 Verona (IT)

(74) Representative: Filler, Wendy Anne, Dr. et al
Glaxo Wellcome plcGlaxo Wellcome House,Berkeley Avenue
Greenford, Middlesex UB6 0NN
Greenford, Middlesex UB6 0NN (GB)

   


(54) QUINOLINE-2-CARBOXYLIC ACID DERIVATIVE AND ITS USE AS EXCITATORY AMINO ACIDS ANTAGONIST