(19)
(11) EP 0 973 748 A1

(12)

(43) Date of publication:
26.01.2000 Bulletin 2000/04

(21) Application number: 98914379.7

(22) Date of filing: 31.03.1998
(51) International Patent Classification (IPC)7C07D 233/54, C07D 213/32, C07D 261/10, C07C 323/57, C07C 311/29, C07D 213/68, C07D 213/12, C07D 213/64, C07D 405/12, C07D 213/34, A61K 31/44, A61K 31/195, A61K 31/41
(86) International application number:
PCT/US9806/365
(87) International publication number:
WO 9843/963 (08.10.1998 Gazette 1998/40)
(84) Designated Contracting States:
AT BE CH DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE

(30) Priority: 01.04.1997 US 825318

(71) Applicant: AGOURON PHARMACEUTICALS, INC.
La Jolla, CA 92037-1022 (US)

(72) Inventors:
  • BENDER, Steven, L.
    Oceanside, CA 92054 (US)
  • ABREO, Melwyn, A.
    Imperial Beach, CA 91932 (US)

(74) Representative: Grünecker, Kinkeldey, Stockmair & SchwanhäusserAnwaltssozietät 
Maximilianstrasse 58
80538 München
80538 München (DE)

   


(54) METALLOPROTEINASE INHIBITORS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR PHARMACEUTICAL USES